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3OTS

MDR769 HIV-1 protease complexed with MA/CA hepta-peptide

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues28
DetailsBINDING SITE FOR CHAIN P OF MA/CA SUBSTRATE PEPTIDE
ChainResidue
AARG8
AHOH239
BARG8
BLEU23
BASN25
BGLY27
BALA28
BASP29
BARG41
BLEU46
BILE47
AASN25
BGLY48
BALA82
BHOH274
BHOH280
PHOH237
PHOH241
PHOH268
PHOH277
PHOH282
AGLY27
AALA28
AASP29
AASP30
AARG41
AVAL84
AHOH172

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Cleavage; by viral protease => ECO:0000250
ChainResidueDetails
PTYR5
BASN25

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine; by host => ECO:0000250
ChainResidueDetails
PTYR5
BPHE99

219869

PDB entries from 2024-05-15

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