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3OMP

Fragment-Based Design of novel Estrogen Receptor Ligands

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE W14 A 1
ChainResidue
ALEU298
ALEU301
AALA302
AGLU305
ALEU339
APHE356
AILE373
AGLY472

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE W14 B 1
ChainResidue
BLEU301
BALA302
BGLU305
BLEU339
BMET340
BILE373
BGLY472
BLEU298

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
CSER13
DSER13

219140

PDB entries from 2024-05-01

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