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3ISN

Crystal structure of HIV-1 RT bound to A 6-vinylpyrimidine inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
C0003676molecular_functionnucleic acid binding
C0003964molecular_functionRNA-directed DNA polymerase activity
C0004523molecular_functionRNA-DNA hybrid ribonuclease activity
C0006278biological_processRNA-templated DNA biosynthetic process
D0003964molecular_functionRNA-directed DNA polymerase activity
D0006278biological_processRNA-templated DNA biosynthetic process
Functional Information from PDB Data
site_idAC1
Number of Residues9
DetailsBINDING SITE FOR RESIDUE EDM C 561
ChainResidue
CMET184
CASP186
CMET230
CGLY231
CLYS263
CTRP266
CHOH578
CHOH631
CHOH672

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING:
ChainResidueDetails
DASP110
DASP185
DASP186

site_idSWS_FT_FI2
Number of Residues2
DetailsSITE: Essential for RT p66/p51 heterodimerization
ChainResidueDetails
DTRP401
DTRP414
CASP498
CASP549

site_idSWS_FT_FI3
Number of Residues2
DetailsSITE: Essential for RT p66/p51 heterodimerization
ChainResidueDetails
CTRP401
CTRP414

site_idSWS_FT_FI4
Number of Residues1
DetailsSITE: Cleavage; by viral protease; partial
ChainResidueDetails
CPHE440

site_idSWS_FT_FI5
Number of Residues1
DetailsSITE: Cleavage; by viral protease => ECO:0000250
ChainResidueDetails
CLEU560

219869

PDB entries from 2024-05-15

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