Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 22 |
Details | BINDING SITE FOR RESIDUE IK2 A 1445 |
Chain | Residue |
A | ARG54 |
A | GLY174 |
A | GLU220 |
A | ASP253 |
A | VAL255 |
A | MET256 |
A | LYS280 |
A | HOH2056 |
A | HOH2115 |
A | HOH2117 |
A | HOH2237 |
A | ILE56 |
B | ALA312 |
B | GLY313 |
B | THR314 |
A | TYR89 |
A | SER144 |
A | GLY145 |
A | THR146 |
A | ASN149 |
A | TYR172 |
A | HIS173 |
site_id | AC2 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE EDO B 1446 |
Chain | Residue |
B | ASP33 |
B | ASN34 |
B | TYR82 |
B | EDO1448 |
site_id | AC3 |
Number of Residues | 23 |
Details | BINDING SITE FOR RESIDUE IK2 B 1447 |
Chain | Residue |
A | ALA312 |
A | GLY313 |
A | THR314 |
A | HOH2113 |
A | HOH2114 |
A | HOH2190 |
B | ARG54 |
B | ILE56 |
B | SER144 |
B | GLY145 |
B | THR146 |
B | ASN149 |
B | TYR172 |
B | HIS173 |
B | GLY174 |
B | GLU220 |
B | ASP253 |
B | VAL255 |
B | MET256 |
B | LYS280 |
B | EDO1453 |
B | HOH2057 |
B | HOH2087 |
site_id | AC4 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EDO B 1448 |
Chain | Residue |
B | HIS80 |
B | ALA81 |
B | TYR82 |
B | LEU403 |
B | GLY406 |
B | EDO1446 |
B | HOH2029 |
site_id | AC5 |
Number of Residues | 24 |
Details | BINDING SITE FOR RESIDUE IK2 C 1445 |
Chain | Residue |
C | ARG54 |
C | ILE56 |
C | TYR89 |
C | SER144 |
C | GLY145 |
C | THR146 |
C | ASN149 |
C | TYR172 |
C | HIS173 |
C | GLY174 |
C | GLU220 |
C | ASP253 |
C | VAL255 |
C | MET256 |
C | LYS280 |
C | ALA312 |
C | GLY313 |
C | THR314 |
C | EDO1449 |
C | HOH2094 |
C | HOH2096 |
C | HOH2097 |
C | HOH2127 |
C | HOH2223 |
site_id | AC6 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO B 1449 |
Chain | Residue |
B | PRO230 |
B | GLU232 |
B | ILE381 |
B | HOH2134 |
B | HOH2160 |
site_id | AC7 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO C 1446 |
Chain | Residue |
C | ALA81 |
C | TYR82 |
C | LEU403 |
C | ARG404 |
C | HOH2044 |
site_id | AC8 |
Number of Residues | 3 |
Details | BINDING SITE FOR RESIDUE EDO C 1447 |
Chain | Residue |
C | ALA180 |
C | GLY226 |
C | ALA384 |
site_id | AC9 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO A 1446 |
Chain | Residue |
A | HIS40 |
A | ARG43 |
A | HOH2238 |
B | GLU120 |
B | ALA123 |
site_id | BC1 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EDO B 1450 |
Chain | Residue |
B | LEU113 |
B | ASN114 |
B | ASN318 |
B | ILE319 |
B | LEU320 |
B | HOH2043 |
A | GLY285 |
site_id | BC2 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO C 1448 |
Chain | Residue |
C | ILE56 |
C | TYR172 |
C | ALA225 |
C | EDO1449 |
C | HOH2112 |
site_id | BC3 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EDO C 1449 |
Chain | Residue |
C | ILE56 |
C | TYR89 |
C | ALA225 |
C | MET256 |
C | LYS280 |
C | IK21445 |
C | EDO1448 |
site_id | BC4 |
Number of Residues | 8 |
Details | BINDING SITE FOR RESIDUE EDO A 1447 |
Chain | Residue |
A | LEU124 |
A | GLU127 |
A | ALA128 |
A | HIS326 |
A | HOH2101 |
A | HOH2193 |
C | ARG43 |
C | GLU120 |
site_id | BC5 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EDO B 1451 |
Chain | Residue |
A | GLU127 |
A | CYS130 |
A | HOH2100 |
A | HOH2109 |
B | ARG46 |
B | HOH2161 |
C | ARG43 |
site_id | BC6 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EDO C 1450 |
Chain | Residue |
A | THR330 |
A | HOH2193 |
A | HOH2195 |
C | ALA67 |
C | VAL77 |
C | GLU120 |
C | HOH2224 |
site_id | BC7 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE EDO A 1448 |
Chain | Residue |
A | PRO221 |
A | PRO230 |
A | ALA231 |
A | LEU236 |
A | LEU269 |
A | LEU368 |
site_id | BC8 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO C 1451 |
Chain | Residue |
A | HOH2093 |
B | ALA67 |
C | HIS326 |
C | THR330 |
C | GLN331 |
site_id | BC9 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO C 1452 |
Chain | Residue |
C | PRO221 |
C | PRO230 |
C | ALA231 |
C | LEU236 |
C | LEU269 |
site_id | CC1 |
Number of Residues | 10 |
Details | BINDING SITE FOR RESIDUE EDO A 1449 |
Chain | Residue |
A | ASN84 |
A | GLY87 |
A | GLU88 |
A | GLY92 |
A | GLY95 |
A | HIS96 |
A | SER418 |
A | HOH2052 |
B | ASN114 |
B | SER116 |
site_id | CC2 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE EDO B 1452 |
Chain | Residue |
B | ALA180 |
B | GLY226 |
B | ALA384 |
B | HOH2071 |
site_id | CC3 |
Number of Residues | 6 |
Details | BINDING SITE FOR RESIDUE EDO B 1453 |
Chain | Residue |
B | ILE56 |
B | TYR89 |
B | ALA225 |
B | MET256 |
B | LYS280 |
B | IK21447 |
site_id | CC4 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE EDO C 1453 |
Chain | Residue |
C | ASN198 |
C | ASP199 |
C | ARG382 |
C | HOH2120 |
C | HOH2122 |
site_id | CC5 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE EDO A 1450 |
Chain | Residue |
A | ASP33 |
A | ASN34 |
A | TYR82 |
A | HOH2228 |