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2L60

A novel design concept: New Y-receptor agonists with increased membrane recruitment, Y2 affinity and selectivity

Functional Information from GO Data
ChainGOidnamespacecontents
A0005179molecular_functionhormone activity
A0005576cellular_componentextracellular region
Functional Information from PROSITE/UniProt
site_idPS00265
Number of Residues17
DetailsPANCREATIC_HORMONE_1 Pancreatic hormone family signature. YyasLrhYlnlVtRqRY
ChainResidueDetails
ATYR24-TYR40

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0000250|UniProtKB:P68005
ChainResidueDetails
ASER17

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Tyrosine amide => ECO:0000269|PubMed:2587421, ECO:0000269|PubMed:3202875
ChainResidueDetails
ATYR40

218853

PDB entries from 2024-04-24

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