Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

1QB6

BOVINE TRYPSIN 3,3'-[3,5-DIFLUORO-4-METHYL-2, 6-PYRIDINEDIYLBIS(OXY)]BIS(BENZENECARBOXIMIDAMIDE) (ZK-805623) COMPLEX

Functional Information from GO Data
ChainGOidnamespacecontents
A0004175molecular_functionendopeptidase activity
A0004252molecular_functionserine-type endopeptidase activity
A0005515molecular_functionprotein binding
A0005576cellular_componentextracellular region
A0005615cellular_componentextracellular space
A0006508biological_processproteolysis
A0007586biological_processdigestion
A0008233molecular_functionpeptidase activity
A0008236molecular_functionserine-type peptidase activity
A0016787molecular_functionhydrolase activity
A0046872molecular_functionmetal ion binding
A0097180cellular_componentserine protease inhibitor complex
A0097655molecular_functionserpin family protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 301
ChainResidue
AGLU58
AASN60
AVAL63
AGLU68
AHOH308
AHOH333

site_idAC2
Number of Residues2
DetailsBINDING SITE FOR RESIDUE K A 302
ChainResidue
AGLN180
ASER183

site_idAC3
Number of Residues14
DetailsBINDING SITE FOR RESIDUE 623 A 300
ChainResidue
ATHR86
ALEU87
ASER114
ACYS115
ASER117
AASP177
ASER178
AGLN180
ATRP199
AGLY200
AGLY202
AGLY210
AHOH444
AASN85

Functional Information from PROSITE/UniProt
site_idPS00134
Number of Residues6
DetailsTRYPSIN_HIS Serine proteases, trypsin family, histidine active site. VSAAHC
ChainResidueDetails
AVAL42-CYS47

site_idPS00135
Number of Residues12
DetailsTRYPSIN_SER Serine proteases, trypsin family, serine active site. DScqGDSGGPVV
ChainResidueDetails
AASP177-VAL188

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsACT_SITE: Charge relay system
ChainResidueDetails
AGLN69
ATHR113
ALYS206

site_idSWS_FT_FI2
Number of Residues7
DetailsBINDING:
ChainResidueDetails
ASER81
AASN83
ATHR86
AILE91
AGLY200
ACYS203
ALYS206

218853

PDB entries from 2024-04-24

PDB statisticsPDBj update infoContact PDBjnumon