1HPV
CRYSTAL STRUCTURE OF HIV-1 PROTEASE IN COMPLEX WITH VX-478, A POTENT AND ORALLY BIOAVAILABLE INHIBITOR OF THE ENZYME
Experimental procedure
Spacegroup name | P 61 |
Unit cell lengths | 63.400, 63.400, 83.800 |
Unit cell angles | 90.00, 90.00, 120.00 |
Refinement procedure
Resolution | 8.000 - 1.900 |
R-factor | 0.192 |
Rwork | 0.192 |
RMSD bond length | 0.011 |
RMSD bond angle | 1.950 |
Phasing software | X-PLOR |
Refinement software | X-PLOR |
Data quality characteristics
Overall | |
High resolution limit [Å] | 1.900 * |
Rmerge | 0.071 * |
Total number of observations | 44734 * |
Number of reflections | 11037 |
Crystallization Conditions
crystal ID | method | pH | temperature | details |
1 |