PDBID: | 8udy | Status: | HPUB -- hold until publication | Title: | Crystal structure of SARS-CoV-2 3CL protease with inhibitor DH-24B | Authors: | Forouhar, F., Liu, H., Zack, A., Iketani, S., Williams, A., Vaz, D.R., Habashi, D.L., Resnick, S.J., Chavez, A., Ho, D.D., Stockwell, B.R. | Deposition date: | 2023-09-29 | Sequence: | >Entity 1 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
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PDBID: | 8qo6 | Status: | HPUB -- hold until publication | Title: | OPR3 variant R283D in complex with NADH4 | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-28 | Release date: | 2025-03-28 | Sequence: | >Entity 1 HHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPDYVAYGQTEAGRLGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qo7 | Status: | HPUB -- hold until publication | Title: | OPR3 variant R283E in complex with NADPH4 | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-28 | Release date: | 2025-03-28 | Sequence: | >Entity 1 HHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPEYVAYGQTEAGRLGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qo8 | Status: | HPUB -- hold until publication | Title: | OPR3 variant R283E in complex with NADH4 | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-28 | Release date: | 2025-03-28 | Sequence: | >Entity 1 HHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPEYVAYGQTEAGRLGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8udf | Status: | HPUB -- hold until publication | Title: | Crystal structure of SARS-CoV-2 3CL protease with inhibitor DEL_7 | Authors: | Forouhar, F., Liu, H., Zack, A., Iketani, S., Williams, A., Vaz, D.R., Habashi, D.L., Resnick, S.J., Chavez, A., Ho, D.D., Stockwell, B.R. | Deposition date: | 2023-09-28 | Sequence: | >Entity 1 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGS(CSO)GSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
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PDBID: | 8udj | Status: | HPUB -- hold until publication | Title: | Crystal structure of SARS-CoV-2 3CL protease with inhibitor DEL_2 | Authors: | Forouhar, F., Liu, H., Zack, A., Iketani, S., Williams, A., Vaz, D.R., Habashi, D.L., Resnick, S.J., Chavez, A., Ho, D.D., Stockwell, B.R. | Deposition date: | 2023-09-28 | Sequence: | >Entity 1 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
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PDBID: | 8udm | Status: | HPUB -- hold until publication | Title: | Crystal structure of SARS-CoV-2 3CL protease with inhibitor ADW-25 | Authors: | Forouhar, F., Liu, H., Zack, A., Iketani, S., Williams, A., Vaz, D.R., Habashi, D.L., Resnick, S.J., Chavez, A., Ho, D.D., Stockwell, B.R. | Deposition date: | 2023-09-28 | Sequence: | >Entity 1 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGS(CSO)GSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
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PDBID: | 8udp | Status: | HPUB -- hold until publication | Title: | Crystal structure of SARS-CoV-2 3CL protease with inhibitor DV-6-4 | Authors: | Forouhar, F., Liu, H., Zack, A., Iketani, S., Williams, A., Vaz, D.R., Habashi, D.L., Resnick, S.J., Chavez, A., Ho, D.D., Stockwell, B.R. | Deposition date: | 2023-09-28 | Sequence: | >Entity 1 SGFRKMAFPSGKVEGCMVQVTCGTTTLNGLWLDDVVYCPRHVICTSEDMLNPNYEDLLIRKSNHNFLVQAGNVQLRVIGHSMQNCVLKLKVDTANPKTPKYKFVRIQPGQTFSVLACYNGSPSGVYQCAMRPNFTIKGSFLNGSCGSVGFNIDYDCVSFCYMHHMELPTGVHAGTDLEGNFYGPFVDRQTAQAAGTDTTITVNVLAWLYAAVINGDRWFLNRFTTTLNDFNLVAMKYNYEPLTQDHVDILGPLSAQTGIAVLDMCASLKELLQNGMNGRTILGSALLEDEFTPFDVVRQCSGVTFQ
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PDBID: | 8qnk | Status: | HPUB -- hold until publication | Title: | OPR3 variant R283D in complex with NADPH4 | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-27 | Release date: | 2025-03-27 | Sequence: | >Entity 1 HHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPDYVAYGQTEAGRLGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qnm | Status: | HPUB -- hold until publication | Title: | OPR3 with redesigned Loop 6 (9aa) in complex with NADPH4 | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-27 | Release date: | 2025-03-27 | Sequence: | >Entity 1 MASHHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPRSDKGGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qnp | Status: | HPUB -- hold until publication | Title: | OPR3 with redesigned loop 6 (9aa) in complex with NADH4 | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-27 | Release date: | 2025-03-27 | Sequence: | >Entity 1 MASHHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPRSDKGGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qnw | Status: | HPUB -- hold until publication | Title: | OPR3 variant with redesigned loop 6 (8aa) | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-27 | Release date: | 2025-03-27 | Sequence: | >Entity 1 MASHHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPGDGRGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qnx | Status: | HPUB -- hold until publication | Title: | OPR3 variant with redesigned loop 6 (8aa) in complex with NADH4 | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-27 | Release date: | 2025-03-27 | Sequence: | >Entity 1 MASHHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPGDGRGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qny | Status: | HPUB -- hold until publication | Title: | OPR3 variant with redesigned loop 6 (8aa) in complex with NADPH4 | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-27 | Release date: | 2025-03-27 | Sequence: | >Entity 1 MASHHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPGDGRGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qn9 | Status: | HPUB -- hold until publication | Title: | OPR3 variant - R283E | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-26 | Release date: | 2025-03-26 | Sequence: | >Entity 1 HHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPEYVAYGQTEAGRLGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qna | Status: | HPUB -- hold until publication | Title: | OPR3 variant - R366A | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-26 | Release date: | 2025-03-26 | Sequence: | >Entity 1 HHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPRYVAYGQTEAGRLGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNAKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qne | Status: | HPUB -- hold until publication | Title: | OPR3 variant with redesigned loop 6 (9aa) | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-26 | Release date: | 2025-03-26 | Sequence: | >Entity 1 MASHHHHHHMASSAQDGNNPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPRSDKGGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFLQGNGSNGPLSRL
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PDBID: | 8qn1 | Status: | HPUB -- hold until publication | Title: | OPR3 variant - R283D | Authors: | Bijelic, A., Macheroux, P., Kerschbaumer, B. | Deposition date: | 2023-09-25 | Sequence: | >Entity 1 NPLFSPYKMGKFNLSHRVVLAPMTRCRALNNIPQAALGEYYEQRATAGGFLITEGTMISPTSAGFPHVPGIFTKEQVREWKKIVDVVHAKGAVIFCQLWHVGRASHEVYQPAGAAPISSTEKPISNRWRILMPDGTHGIYPKPRAIGTYEISQVVEDYRRSALNAIEAGFDGIEIHGAHGYLIDQFLKDGINDRTDEYGGSLANRCKFITQVVQAVVSAIGADRVGVRVSPAIDHLDAMDSNPLSLGLAVVERLNKIQLHSGSKLAYLHVTQPDYVAYGQTEAGRLGSEEEEARLMRTLRNAYQGTFICSGGYTRELGIEAVAQGDADLVSYGRLFISNPDLVMRIKLNAPLNKYNRKTFYTQDPVVGYTDYPFL
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PDBID: | 8ubq | Status: | HPUB -- hold until publication | Title: | EcDsbA soaked with N-(2-fluorophenyl)-5-methylisoxazole-3-carboxamide and 2-benzyl-4-phenylthiazole-5-carboxylic acid | Authors: | Wang, G., Heras, B. | Deposition date: | 2023-09-24 | Sequence: | >Entity 1 AQYEDGKQYTTLEKPVAGAPQVLEFFSFFCPHCYQFEEVLHISDNVKKKLPEGVKMTKYHVNFMGGDLGKDLTQAWAVAMALGVEDKVTVPLFEGVQKTQTIRSASDIRDVFINAGIKGEEYDAAWNSFVVKSLVAQQEKAAADVQLRGVPAMFVNGKYQLNPQGMDTSNMDVFVQQYADTVKYLSEKK
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PDBID: | 8uaw | Status: | HPUB -- hold until publication | Title: | Cryo-EM Structure of Brucella Abortus Lumazine Synthase (BLS) Engineered with Shiga Toxin II subunit B (Stx2B) | Authors: | Cristofalo, A.E., Sharma, A., Cerutti, M.L., Sharma, K., Zylberman, V., Goldbaum, F.A., Borgnia, M.J., Otero, L.H. | Deposition date: | 2023-09-22 |
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PDBID: | 8ub5 | Status: | HPUB -- hold until publication | Title: | The Apo NanH structure from Clostridium perfringens | Authors: | Medley, B.J., Boraston, A.B. | Deposition date: | 2023-09-22 |
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PDBID: | 8qmb | Status: | HPUB -- hold until publication | Title: | Nucleant-assisted 2.0 A resolution structure of the Streptococcus pneumoniae topoisomerase IV-V18mer DNA complex with the novel fluoroquinolone Delafloxacin | Authors: | Najmudin, S., Pan, X.S., Wang, B., Chayen, N.E., Fisher, L.M., Sanderson, M.R. | Deposition date: | 2023-09-21 |
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PDBID: | 8qmc | Status: | HOLD -- hold until a certain date | Title: | High resolution structure of the Streptococcus pneumoniae topoisomerase IV-complex with the V-site 18mer dsDNA and novel fluoroquinolone Delafloxacin | Authors: | Najmudin, S., Pan, X.S., Wang, B., Chayen, N.E., Fisher, L.M., Sanderson, M.R. | Deposition date: | 2023-09-21 | Release date: | 2024-09-21 |
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PDBID: | 8qkv | Status: | HOLD -- hold until a certain date | Title: | SWR1-nucleosome complex in configuration 2 | Authors: | Jalal, A.S.B., Wigley, D.B. | Deposition date: | 2023-09-18 | Release date: | 2024-09-18 |
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PDBID: | 8qku | Status: | HOLD -- hold until a certain date | Title: | SWR1-nucleosome complex in configuration 1 | Authors: | Jalal, A.S.B., Wigley, D.B. | Deposition date: | 2023-09-18 | Release date: | 2024-09-18 |
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