PDBID: | 8r0q | Status: | HPUB -- hold until publication | Title: | Pim1 in complex with 6-bromo-1H-benzo[d]imidazol-2-amine and Pimtide | Authors: | Hochban, P.M.M., Heine, A., Diederich, W.E. | Deposition date: | 2023-10-31 | Sequence: | >Entity 1 SMLLSKINSLAHLRAAPCNDLHATKLAPGKEKEPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVS(SEP)ECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLSPGPS
>Entity 2 ARKRRRHPSGPPTA
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PDBID: | 8r0t | Status: | HOLD -- hold until a certain date | Deposition date: | 2023-10-31 | Release date: | 2024-10-31 |
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PDBID: | 8r0w | Status: | HPUB -- hold until publication | Title: | Pim1 in complex with 5-bromobenzo[d]oxazol-2-amine and Pimtide | Authors: | Hochban, P.M.M., Heine, A., Diederich, W.E. | Deposition date: | 2023-11-01 | Sequence: | >Entity 1 SMLLSKINSLAHLRAAPCNDLHATKLAPGKEKEPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVS(SEP)ECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLSPGPS
>Entity 2 ARKRRRHPSGPPTA
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PDBID: | 8r0y | Status: | HPUB -- hold until publication | Title: | Pim1 in complex with 3-((3-hydroxyphenyl)amino)quinoxaline-2-carboxylic acid and Pimtide | Authors: | Hochban, P.M.M., Heine, A., Diederich, W.E. | Deposition date: | 2023-11-01 | Sequence: | >Entity 1 SMLLSKINSLAHLRAAPCNDLHATKLAPGKEKEPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVS(SEP)ECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLSPGPS
>Entity 2 ARKRRRHPSGPPTA
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PDBID: | 8r13 | Status: | AUTH -- processed, waiting for author review and approval | Title: | Alpha-1-antitrypsin (Met374Phe) in the native conformation | Authors: | Aldobiyan, I., Lomas, D.A., Irving, J.A. | Deposition date: | 2023-11-01 |
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PDBID: | 8r1b | Status: | AUTH -- processed, waiting for author review and approval | Deposition date: | 2023-11-01 |
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PDBID: | 8r1e | Status: | HPUB -- hold until publication | Title: | crystal structure of acyl-CoA dehydrogenase FadE2 mutant (PA0508 M130G E296A Q303A) from Pseudomonas aeruginosa | Authors: | Wang, M., Brear, P., Welch, M. | Deposition date: | 2023-11-01 |
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PDBID: | 8r1k | Status: | HPUB -- hold until publication | Title: | Pim1 in complex with 6-bromobenzo[d]oxazol-2-amine and Pimtide | Authors: | Hochban, P.M.M., Heine, A., Diederich, W.E. | Deposition date: | 2023-11-02 | Sequence: | >Entity 1 SMLLSKINSLAHLRAAPCNDLHATKLAPGKEKEPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVS(SEP)ECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLSPGPS
>Entity 2 ARKRRRHPSGPPTA
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PDBID: | 8r1q | Status: | HOLD -- hold until a certain date | Title: | SARS-CoV-2 Mpro (Omicron, P132H+T169S) in complex with alpha-ketoamide 13b-K | Authors: | Sun, X., Ibrahim, M., Hilgenfeld, R. | Deposition date: | 2023-11-02 | Release date: | 2023-11-30 |
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PDBID: | 8r1r | Status: | AUTH -- processed, waiting for author review and approval | Deposition date: | 2023-11-02 | Release date: | 2024-11-02 |
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PDBID: | 8r1s | Status: | HOLD -- hold until a certain date | Deposition date: | 2023-11-02 | Release date: | 2025-05-06 |
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PDBID: | 8r1u | Status: | HPUB -- hold until publication | Deposition date: | 2023-11-02 |
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PDBID: | 8r1w | Status: | HPUB -- hold until publication | Title: | Pim1 in complex with 4-(5-(4-aminophenyl)-2H-1,2,3-triazol-4-yl)benzoic acid and Pimtide | Authors: | Hochban, P.M.M., Heine, A., Diederich, W.E. | Deposition date: | 2023-11-02 | Sequence: | >Entity 1 SMLLSKINSLAHLRAAPCNDLHATKLAPGKEKEPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVS(SEP)ECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLSPGPS
>Entity 2 ARKRRRHPSGPPTA
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PDBID: | 8r1z | Status: | HPUB -- hold until publication | Deposition date: | 2023-11-02 |
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PDBID: | 8r21 | Status: | HPUB -- hold until publication | Title: | Alpha-1-antitrypsin (Ile340Trp) in the native conformation | Authors: | Aldobiyan, I., Lee, H.J., Lomas, D.A., Irving, J.A. | Deposition date: | 2023-11-02 | Sequence: | >Entity 1 MRGSHHHHHHTDPQGDAAQKTDTSHHDQDHPTFNKITPNLAEFAFSLYRQLAHQSNSTNIFFSPVSIATAFAMLSLGTKADTHDEILEGLNFNLTEIPEAQIHEGFQELLRTLNQPDSQLQLTTGNGLFLSEGLKLVDKFLEDVKKLYHSEAFTVNFGDTEEAKKQINDYVEKGTQGKIVDLVKELDRDTVFALVNYIFFKGKWERPFEVKDTEEEDFHVDQVTTVKVPMMKRLGMFNIQHCKKLSSWVLLMKYLGNATAIFFLPDEGKLQHLENELTHDIITKFLENEDRRSASLHLPKLSITGTYDLKSVLGQLGITKVFSNGADLSGVTEEAPLKLSKAVHKAVLTWDEKGTEAAGAMFLEAIPMSIPPEVKFNKPFVFLMIEQNTKSPLFMGKVVNPTQK
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PDBID: | 8r24 | Status: | HOLD -- hold until a certain date | Title: | SARS-CoV-2 Mpro (Omicron, P132H+T169S) free enzyme | Authors: | Sun, X., Ibrahim, M., El Kilani, H., Hilgenfeld, R. | Deposition date: | 2023-11-02 | Release date: | 2023-11-30 |
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PDBID: | 8r25 | Status: | HPUB -- hold until publication | Title: | Pim1 in complex with 4-(5-(4-aminophenyl)-1H-pyrazol-1-yl)benzoic acid and Pimtide | Authors: | Hochban, P.M.M., Heine, A., Diederich, W.E. | Deposition date: | 2023-11-03 | Sequence: | >Entity 1 SMLLSKINSLAHLRAAPCNDLHATKLAPGKEKEPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVS(SEP)ECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLSPGPS
>Entity 2 ARKRRRHPSGPPTA
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PDBID: | 8r26 | Status: | HOLD -- hold until a certain date | Title: | SARS-CoV-2 Mpro (Omicron,P132H) in complex with alpha-ketoamide 13b-K at pH 8.5 | Authors: | Ibrahim, M., Sun, X., Hilgenfeld, R. | Deposition date: | 2023-11-03 | Release date: | 2023-12-01 |
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PDBID: | 8r27 | Status: | HPUB -- hold until publication | Title: | Pim1 in complex with (Z)-4-(1-cyano-2-(4-hydroxyphenyl)vinyl)benzoic acid and Pimtide | Authors: | Hochban, P.M.M., Heine, A., Diederich, W.E. | Deposition date: | 2023-11-03 | Sequence: | >Entity 1 SMLLSKINSLAHLRAAPCNDLHATKLAPGKEKEPLESQYQVGPLLGSGGFGSVYSGIRVSDNLPVAIKHVEKDRISDWGELPNGTRVPMEVVLLKKVSSGFSGVIRLLDWFERPDSFVLILERPEPVQDLFDFITERGALQEELARSFFWQVLEAVRHCHNCGVLHRDIKDENILIDLNRGELKLIDFGSGALLKDTVYTDFDGTRVYSPPEWIRYHRYHGRSAAVWSLGILLYDMVCGDIPFEHDEEIIGGQVFFRQRVS(SEP)ECQHLIRWCLALRPSDRPTFEEIQNHPWMQDVLLPQETAEIHLHSLSPGPS
>Entity 2 ARKRRRHPSGPPTA
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PDBID: | 8r28 | Status: | HPUB -- hold until publication | Deposition date: | 2023-11-03 |
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PDBID: | 8r29 | Status: | HPUB -- hold until publication | Title: | Crystal structure of domain swapped dimer of Amacstatin-2, a cystatin from the hard tick Amblyomma maculatum | Authors: | Busa, M., Mares, M. | Deposition date: | 2023-11-03 |
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PDBID: | 8r2a | Status: | HPUB -- hold until publication | Title: | CpKRS complexed with lysine and an inhibitor | Authors: | Dawson, A., Baragana, B., Caldwell, N. | Deposition date: | 2023-11-03 |
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PDBID: | 8r2f | Status: | HPUB -- hold until publication | Title: | human carbonic anhydrase II in complex with 4-(((dimethoxyphosphoryl)(4-((dimethoxyphosphoryl)((4-sulfamoylphenyl)amino)methyl)phenyl)methyl)amino)phenyl sulfuramidite | Authors: | Angeli, A., Ferraroni, M. | Deposition date: | 2023-11-04 | Sequence: | >Entity 1 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK
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PDBID: | 8r2k | Status: | HPUB -- hold until publication | Title: | Human Carbonic Anhydrase II in complex with 4-((2-oxo-5-(3,4,5-trimethoxyphenyl)-2,5-dihydrofuran-3-yl)amino)benzenesulfonamide | Authors: | Angeli, A., Ferraroni, M. | Deposition date: | 2023-11-06 | Sequence: | >Entity 1 MSHHWGYGKHNGPEHWHKDFPIAKGERQSPVDIDTHTAKYDPSLKPLSVSYDQATSLRILNNGHAFNVEFDDSQDKAVLKGGPLDGTYRLIQFHFHWGSLDGQGSEHTVDKKKYAAELHLVHWNTKYGDFGKAVQQPDGLAVLGIFLKVGSAKPGLQKVVDVLDSIKTKGKSADFTNFDPRGLLPESLDYWTYPGSLTTPPLLECVTWIVLKEPISVSSEQVLKFRKLNFNGEGEPEELMVDNWRPAQPLKNRQIKASFK
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PDBID: | 8r2n | Status: | AUTH -- processed, waiting for author review and approval | Title: | Structure of the BeeR filament | Authors: | Bergeron, J.R.C., Kollman, J.M. | Deposition date: | 2023-11-07 |
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