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PDB: 1 results
3MBL
Crystal Structure of the human mitogen-activated protein kinase kinase 1 (MEK 1) in complex with ligand and MgADP
Descriptor:
5-acetyl-2-[(2-fluoro-4-iodophenyl)amino]-N-(2-hydroxyethoxy)-1-methyl-1H-pyrrole-3-carboxamide, ADENOSINE-5'-DIPHOSPHATE, Dual specificity mitogen-activated protein kinase kinase 1, ...
Authors:
Dougan, D.R
,
Mol, C.D.
Deposit date:
2010-03-25
Release date:
2010-07-28
Last modified:
2024-02-21
Method:
X-RAY DIFFRACTION (2.6 Å)
Cite:
Structure-based design and synthesis of pyrrole derivatives as MEK inhibitors.
Bioorg.Med.Chem.Lett., 20, 2010
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數據於2024-05-15公開中