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PDB: 1 件

6K9U
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Discovery of Pyrazolo[1,5-a]pyrimidine Derivative as a Highly Selective PDE10A Inhibitor
分子名称: 2-(3,7-dimethylquinoxalin-2-yl)-~{N}-(oxan-4-yl)-5-pyrrolidin-1-yl-pyrazolo[1,5-a]pyrimidin-7-amine, MAGNESIUM ION, SULFATE ION, ...
著者Takedomi, K, Koizumi, Y.
登録日2019-06-18
公開日2019-07-17
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Discovery of a pyrazolo[1,5-a]pyrimidine derivative (MT-3014) as a highly selective PDE10A inhibitor via core structure transformation from the stilbene moiety.
Bioorg.Med.Chem., 27, 2019

220113

件を2024-05-22に公開中

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