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PDB: 2 results
6PGO
Crystal structure of human KRAS G12C covalently bound to a phthalazine inhibitor
Descriptor:
1-{4-[7-chloro-6-(2-fluoro-6-hydroxyphenyl)-4-phenylphthalazin-1-yl]piperazin-1-yl}propan-1-one, GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:
Mohr, C.
Deposit date:
2019-06-24
Release date:
2019-12-25
Last modified:
2020-01-22
Method:
X-RAY DIFFRACTION (1.6 Å)
Cite:
Discovery of a Covalent Inhibitor of KRASG12C(AMG 510) for the Treatment of Solid Tumors.
J.Med.Chem., 63, 2020
6PGP
Crystal structure of human KRAS G12C covalently bound to a quinazolinone inhibitor
Descriptor:
6-chloro-7-(2-fluoro-6-hydroxyphenyl)-4-(4-propanoylpiperazin-1-yl)-1-[2-(propan-2-yl)phenyl]quinazolin-2(1H)-one, CALCIUM ION, GTPase KRas, ...
Authors:
Mohr, C
,
Whittington, D.A.
Deposit date:
2019-06-24
Release date:
2019-12-25
Last modified:
2020-01-22
Method:
X-RAY DIFFRACTION (1.5 Å)
Cite:
Discovery of a Covalent Inhibitor of KRASG12C(AMG 510) for the Treatment of Solid Tumors.
J.Med.Chem., 63, 2020
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數據於2024-08-14公開中