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PDB: 3 results

8QKE
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BU of 8qke by Molmil
PvSub1 Catalytic Domain in Complex with Peptidomimetic Inhibitor (MH-13)
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Peptidomimetic Inhibitor (MH-13), ...
Authors:Batista, F.A, Martinez, M, Bouillon, A, Mechaly, A, Alzari, P.M, Haouz, A, Barale, J.C.
Deposit date:2023-09-15
Release date:2024-03-20
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (1.504 Å)
Cite:Insights from structure-activity relationships and the binding mode of peptidic alpha-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1.
Eur.J.Med.Chem., 269, 2024
8QKG
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BU of 8qkg by Molmil
PvSub1 Catalytic Domain in Complex with Peptidomimetic Inhibitor (MAM-125)
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Peptidomimetic Inhibitor (MAM-125), ...
Authors:Batista, F.A, Martinez, M, Bouillon, A, Mechaly, A, Alzari, P.M, Haouz, A, Barale, J.C.
Deposit date:2023-09-15
Release date:2024-03-20
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (1.538 Å)
Cite:Insights from structure-activity relationships and the binding mode of peptidic alpha-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1.
Eur.J.Med.Chem., 269, 2024
8QKJ
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BU of 8qkj by Molmil
PvSub1 Catalytic Domain in Complex with Peptidomimetic Inhibitor (MAM-133)
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, Peptidomimetic Inhibitor (MAM-133), ...
Authors:Batista, F.A, Martinez, M, Bouillon, A, Mechaly, A, Alzari, P.M, Haouz, A, Barale, J.C.
Deposit date:2023-09-15
Release date:2024-03-20
Last modified:2024-05-01
Method:X-RAY DIFFRACTION (1.767 Å)
Cite:Insights from structure-activity relationships and the binding mode of peptidic alpha-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1.
Eur.J.Med.Chem., 269, 2024

222036

數據於2024-07-03公開中

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