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PDB: 2 results

4X5Z
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BU of 4x5z by Molmil
menin in complex with MI-136
Descriptor: 1,2-ETHANEDIOL, 5-[(4-{[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]amino}piperidin-1-yl)methyl]-1H-indole-2-carbonitrile, DIMETHYL SULFOXIDE, ...
Authors:Pollock, J, Borkin, D, Cierpicki, T, Grembecka, J.
Deposit date:2014-12-06
Release date:2015-04-15
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.86 Å)
Cite:Pharmacologic Inhibition of the Menin-MLL Interaction Blocks Progression of MLL Leukemia In Vivo.
Cancer Cell, 27, 2015
4X5Y
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BU of 4x5y by Molmil
Menin in complex with MI-503
Descriptor: 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 4-methyl-1-(1H-pyrazol-4-ylmethyl)-5-[(4-{[6-(2,2,2-trifluoroethyl)thieno[2,3-d]pyrimidin-4-yl]amino}piperidin-1-yl)methyl]-1H-indole-2-carbonitrile, ...
Authors:Pollock, J, Borkin, D, Cierpicki, T, Grembecka, J.
Deposit date:2014-12-06
Release date:2015-04-15
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (1.59 Å)
Cite:Pharmacologic Inhibition of the Menin-MLL Interaction Blocks Progression of MLL Leukemia In Vivo.
Cancer Cell, 27, 2015

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數據於2024-07-17公開中

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