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PDB: 2 results
4WSY
Crystal structure of human Pim-1 kinase in complex with a thiazolamine-indazole inhibitor.
Descriptor:
5-[3-(quinolin-3-yl)-2H-indazol-5-yl]-1,3-thiazol-2-amine, GLYCEROL, Serine/threonine-protein kinase pim-1
Authors:
Mohr, C.
Deposit date:
2014-10-28
Release date:
2015-02-11
Last modified:
2023-12-27
Method:
X-RAY DIFFRACTION (2.3 Å)
Cite:
Discovery of 5-(1H-indol-5-yl)-1,3,4-thiadiazol-2-amines as potent PIM inhibitors.
Bioorg.Med.Chem.Lett., 25, 2015
4WT6
Crystal structure of human Pim-1 kinase in complex with a thiadiazolamine-indole inhibitor.
Descriptor:
6-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1H-indol-3-yl]-N-cyclopentylpyridin-2-amine, GLYCEROL, Serine/threonine-protein kinase pim-1
Authors:
Mohr, C.
Deposit date:
2014-10-29
Release date:
2015-02-11
Last modified:
2023-12-27
Method:
X-RAY DIFFRACTION (2.3 Å)
Cite:
Discovery of 5-(1H-indol-5-yl)-1,3,4-thiadiazol-2-amines as potent PIM inhibitors.
Bioorg.Med.Chem.Lett., 25, 2015
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數據於2024-10-16公開中