English
日本語
简体中文
繁體中文
한국어
✖
Menu
RCSB PDB
PDBe
BMRB
Adv. Search
Search help
PDB: 4 results
6V90
Crystal structure of the p300 acetyltransferase domain with AcCoA competitive inhibitor 12
Descriptor:
(2R)-2-{[2-(4-cyanophenyl)ethyl]amino}-N-[5-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-2-phenylacetamide, CHLORIDE ION, Histone acetyltransferase p300, ...
Authors:
Gardberg, A.S.
Deposit date:
2019-12-12
Release date:
2020-04-01
Last modified:
2024-04-03
Method:
X-RAY DIFFRACTION (2.04 Å)
Cite:
Early Drug-Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors.
Chemmedchem, 15, 2020
6V8N
Crystal structure of the p300 acetyltransferase domain with AcCoA competitive inhibitor 17
Descriptor:
(2R)-2-{[(2S)-2-(4-cyanophenyl)propyl]amino}-N-[5-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl]-2-phenylacetamide, CHLORIDE ION, Histone acetyltransferase p300, ...
Authors:
Gardberg, A.S
,
Wilson, J.E.
Deposit date:
2019-12-11
Release date:
2020-04-01
Last modified:
2024-04-03
Method:
X-RAY DIFFRACTION (2.3 Å)
Cite:
Early Drug-Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors.
Chemmedchem, 15, 2020
6V8K
Crystal structure of the p300 acetyltransferase domain with peptide-competitive inhibitor 2
Descriptor:
1-(2-methyl-1H-indol-3-yl)-2-[(2R)-2-methylpiperidin-1-yl]ethan-1-one, COENZYME A, DIMETHYL SULFOXIDE, ...
Authors:
Gardberg, A.S.
Deposit date:
2019-12-11
Release date:
2020-04-01
Last modified:
2024-04-03
Method:
X-RAY DIFFRACTION (1.84 Å)
Cite:
Early Drug-Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors.
Chemmedchem, 15, 2020
6V8B
Crystal structure of the p300 acetyltransferase domain with AcCoA competitive inhibitor 1
Descriptor:
4-(2-{[(1R)-2-(1H-indol-3-yl)-2-oxo-1-phenylethyl]amino}ethyl)benzene-1-sulfonamide, CHLORIDE ION, Histone acetyltransferase p300, ...
Authors:
Gardberg, A.S.
Deposit date:
2019-12-10
Release date:
2020-04-01
Last modified:
2024-04-03
Method:
X-RAY DIFFRACTION (3.13 Å)
Cite:
Early Drug-Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors.
Chemmedchem, 15, 2020
Home
首頁
統計數據
幫助
FAQ
聯絡我們
引用PDBj / 使用條款
相關連接
Settings
數據儲存 (OneDep)
幫助
Deposition to PDB, EMDB or BMRB
下載
下載PDB存檔 / 快照存檔
標準格式
PDBx/mmCIF Resources
格式轉換
PDBx/mmCIF editor
Quick links
幫助
PDB格式不兼容數據
Group Depositions
Chemical Component entries
Latest entries
查詢
幫助
Search PDB (PDBj Mine)
Search PDBj RDB
Chemie search
Search BMRB
Sequence-Navigator
DASH
EM Navigator
Omokage search
Omokage搜索
wwPDB/RDF
RDF Portal
Status search
Molecular Viewers
幫助
jV: Graphic Viewer
Molmil: WebGL Mol. Viewer
服務&軟體
幫助
Yorodumi
ASH
MAFFTash
NMRToolBox
gmfit
CRNPRED
Spanner
SFAS
HOMCOS
衍生資料庫
幫助
eF-site
eF-seek
eF-surf
ProMode Elastic
hGTOP
教材
幫助
eProtS
本月的分子
Previous workshop
Games
Papermodels
關於PDBj
幫助
出版物
新聞發佈 / 公共關係資源
PDBj成員
PDBj諮詢委員會
個人資料保護方針
221051
數據於2024-06-12公開中