5R85
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![BU of 5r85 by Molmil](/molmil-images/mine/5r85) | |
5R86
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![BU of 5r86 by Molmil](/molmil-images/mine/5r86) | |
5R87
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![BU of 5r87 by Molmil](/molmil-images/mine/5r87) | |
5R88
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![BU of 5r88 by Molmil](/molmil-images/mine/5r88) | |
5R89
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![BU of 5r89 by Molmil](/molmil-images/mine/5r89) | |
5R8A
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![BU of 5r8a by Molmil](/molmil-images/mine/5r8a) | PanDDA analysis group deposition INTERLEUKIN-1 BETA -- Fragment Z1492796719 in complex with INTERLEUKIN-1 BETA | Descriptor: | Interleukin-1 beta, SULFATE ION, ~{N}-[(3~{R})-1,2,3,4-tetrahydroquinolin-3-yl]ethanamide | Authors: | De Nicola, G.F, Nichols, C.E. | Deposit date: | 2020-03-03 | Release date: | 2020-04-22 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.47 Å) | Cite: | Mining the PDB for Tractable Cases Where X-ray Crystallography Combined with Fragment Screens Can Be Used to Systematically Design Protein-Protein Inhibitors: Two Test Cases Illustrated by IL1 beta-IL1R and p38 alpha-TAB1 Complexes. J.Med.Chem., 63, 2020
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5R8B
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![BU of 5r8b by Molmil](/molmil-images/mine/5r8b) | PanDDA analysis group deposition INTERLEUKIN-1 BETA -- Fragment Z2027049478 in complex with INTERLEUKIN-1 BETA | Descriptor: | 5-(1,3-thiazol-2-yl)-1H-1,2,4-triazole, Interleukin-1 beta, SULFATE ION | Authors: | De Nicola, G.F, Nichols, C.E. | Deposit date: | 2020-03-03 | Release date: | 2020-04-22 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.49 Å) | Cite: | Mining the PDB for Tractable Cases Where X-ray Crystallography Combined with Fragment Screens Can Be Used to Systematically Design Protein-Protein Inhibitors: Two Test Cases Illustrated by IL1 beta-IL1R and p38 alpha-TAB1 Complexes. J.Med.Chem., 63, 2020
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5R8C
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![BU of 5r8c by Molmil](/molmil-images/mine/5r8c) | |
5R8D
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![BU of 5r8d by Molmil](/molmil-images/mine/5r8d) | |
5R8E
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![BU of 5r8e by Molmil](/molmil-images/mine/5r8e) | PanDDA analysis group deposition INTERLEUKIN-1 BETA -- Fragment Z57475877 in complex with INTERLEUKIN-1 BETA | Descriptor: | Interleukin-1 beta, SULFATE ION, ~{N}-(2-ethyl-1,2,3,4-tetrazol-5-yl)butanamide | Authors: | De Nicola, G.F, Nichols, C.E. | Deposit date: | 2020-03-03 | Release date: | 2020-04-22 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.35 Å) | Cite: | Mining the PDB for Tractable Cases Where X-ray Crystallography Combined with Fragment Screens Can Be Used to Systematically Design Protein-Protein Inhibitors: Two Test Cases Illustrated by IL1 beta-IL1R and p38 alpha-TAB1 Complexes. J.Med.Chem., 63, 2020
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5R8F
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![BU of 5r8f by Molmil](/molmil-images/mine/5r8f) | |
5R8G
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![BU of 5r8g by Molmil](/molmil-images/mine/5r8g) | |
5R8H
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![BU of 5r8h by Molmil](/molmil-images/mine/5r8h) | |
5R8I
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![BU of 5r8i by Molmil](/molmil-images/mine/5r8i) | |
5R8J
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![BU of 5r8j by Molmil](/molmil-images/mine/5r8j) | |
5R8K
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![BU of 5r8k by Molmil](/molmil-images/mine/5r8k) | |
5R8L
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![BU of 5r8l by Molmil](/molmil-images/mine/5r8l) | |
5R8M
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![BU of 5r8m by Molmil](/molmil-images/mine/5r8m) | |
5R8N
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![BU of 5r8n by Molmil](/molmil-images/mine/5r8n) | PanDDA analysis group deposition INTERLEUKIN-1 BETA -- Fragment Z57292400 in complex with INTERLEUKIN-1 BETA | Descriptor: | 3-ethoxy-~{N}-(2-methyl-1,2,3,4-tetrazol-5-yl)benzamide, Interleukin-1 beta, SULFATE ION | Authors: | De Nicola, G.F, Nichols, C.E. | Deposit date: | 2020-03-03 | Release date: | 2020-04-22 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.48 Å) | Cite: | Mining the PDB for Tractable Cases Where X-ray Crystallography Combined with Fragment Screens Can Be Used to Systematically Design Protein-Protein Inhibitors: Two Test Cases Illustrated by IL1 beta-IL1R and p38 alpha-TAB1 Complexes. J.Med.Chem., 63, 2020
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5R8O
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![BU of 5r8o by Molmil](/molmil-images/mine/5r8o) | |
5R8P
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![BU of 5r8p by Molmil](/molmil-images/mine/5r8p) | |
5R8Q
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![BU of 5r8q by Molmil](/molmil-images/mine/5r8q) | |