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PDB: 3 results
3NUY
phosphoinositide-dependent kinase-1 (PDK1) with fragment17
Descriptor:
GLYCEROL, PkB-like, SULFATE ION, ...
Authors:
Campobasso, N
,
Ward, P.
Deposit date:
2010-07-07
Release date:
2011-05-25
Last modified:
2018-10-10
Method:
X-RAY DIFFRACTION (2.1 Å)
Cite:
Aminoindazole PDK1 Inhibitors: A Case Study in Fragment-Based Drug Discovery.
ACS Med Chem Lett, 1, 2010
3NUS
phosphoinositide-dependent kinase-1 (PDK1) with fragment8
Descriptor:
1H-indazol-3-amine, GLYCEROL, SULFATE ION, ...
Authors:
Campobasso, N
,
Ward, P.
Deposit date:
2010-07-07
Release date:
2011-05-25
Last modified:
2018-10-10
Method:
X-RAY DIFFRACTION (2.75 Å)
Cite:
Aminoindazole PDK1 Inhibitors: A Case Study in Fragment-Based Drug Discovery.
ACS Med Chem Lett, 1, 2010
3NUU
phosphoinositide-dependent kinase-1 (PDK1) with fragment11
Descriptor:
3,4-dihydroisoquinolin-1(2H)-one, GLYCEROL, PkB-like, ...
Authors:
Campobasso, N
,
Ward, P.
Deposit date:
2010-07-07
Release date:
2011-05-25
Last modified:
2018-10-10
Method:
X-RAY DIFFRACTION (1.9803 Å)
Cite:
Aminoindazole PDK1 Inhibitors: A Case Study in Fragment-Based Drug Discovery.
ACS Med Chem Lett, 1, 2010
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数据于2024-06-12公开中