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PDB: 1 results

3P9J
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BU of 3p9j by Molmil
Aurora A kinase domain with phthalazinone pyrazole inhibitor
Descriptor: 4-[(5-methyl-1H-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2H)-one, Serine/threonine-protein kinase 6
Authors:Kairies, N.A, Oliveira, T, Engh, R.A.
Deposit date:2010-10-17
Release date:2011-03-23
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of aurora-a kinase.
J.Med.Chem., 54, 2011

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数据于2024-07-10公开中

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