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PDB: 2 results
5KBQ
Pak1 in complex with bis-anilino pyrimidine inhibitor
Descriptor:
Serine/threonine-protein kinase PAK 1, [4-methyl-3-[methyl-[2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]pyrimidin-4-yl]amino]phenyl]methanol
Authors:
Ferguson, A.
Deposit date:
2016-06-03
Release date:
2016-09-28
Last modified:
2023-09-27
Method:
X-RAY DIFFRACTION (2.58 Å)
Cite:
Optimization of Highly Kinase Selective Bis-anilino Pyrimidine PAK1 Inhibitors.
ACS Med Chem Lett, 7, 2016
5KBR
Pak1 in complex with 7-azaindole inhibitor
Descriptor:
(4-chlorophenyl)-[5-(1-piperidin-4-ylpyrazol-4-yl)-1~{H}-pyrrolo[2,3-b]pyridin-3-yl]methanone, Serine/threonine-protein kinase PAK 1
Authors:
Ferguson, A.
Deposit date:
2016-06-03
Release date:
2016-09-28
Last modified:
2023-09-27
Method:
X-RAY DIFFRACTION (2.36 Å)
Cite:
Optimization of Highly Kinase Selective Bis-anilino Pyrimidine PAK1 Inhibitors.
ACS Med Chem Lett, 7, 2016
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数据于2024-07-10公开中