Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 2 results

5KBQ
DownloadVisualize
BU of 5kbq by Molmil
Pak1 in complex with bis-anilino pyrimidine inhibitor
Descriptor: Serine/threonine-protein kinase PAK 1, [4-methyl-3-[methyl-[2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]pyrimidin-4-yl]amino]phenyl]methanol
Authors:Ferguson, A.
Deposit date:2016-06-03
Release date:2016-09-28
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.58 Å)
Cite:Optimization of Highly Kinase Selective Bis-anilino Pyrimidine PAK1 Inhibitors.
ACS Med Chem Lett, 7, 2016
5KBR
DownloadVisualize
BU of 5kbr by Molmil
Pak1 in complex with 7-azaindole inhibitor
Descriptor: (4-chlorophenyl)-[5-(1-piperidin-4-ylpyrazol-4-yl)-1~{H}-pyrrolo[2,3-b]pyridin-3-yl]methanone, Serine/threonine-protein kinase PAK 1
Authors:Ferguson, A.
Deposit date:2016-06-03
Release date:2016-09-28
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (2.36 Å)
Cite:Optimization of Highly Kinase Selective Bis-anilino Pyrimidine PAK1 Inhibitors.
ACS Med Chem Lett, 7, 2016

222415

数据于2024-07-10公开中

PDB statisticsPDBj update infoContact PDBjnumon