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PDB: 2 results

6HJK
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BU of 6hjk by Molmil
Crystal Structure of Aurora-A L210C catalytic domain in complex with ASDO2
Descriptor: (~{E})-~{N}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-but-2-enamide, Aurora kinase A, CHLORIDE ION, ...
Authors:Bayliss, R, McIntyre, P.J.
Deposit date:2018-09-04
Release date:2018-10-03
Last modified:2024-05-15
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Type II Kinase Inhibitors Targeting Cys-Gatekeeper Kinases Display Orthogonality with Wild Type and Ala/Gly-Gatekeeper Kinases.
ACS Chem. Biol., 13, 2018
6HJJ
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BU of 6hjj by Molmil
Crystal structure of Aurora-A L210C catalytic domain in complex with ASDO6 ligand
Descriptor: 2,5,8,11-TETRAOXATRIDECANE, ACETATE ION, Aurora kinase A, ...
Authors:Bayliss, R, McIntyre, P.J.
Deposit date:2018-09-04
Release date:2018-10-03
Last modified:2024-05-15
Method:X-RAY DIFFRACTION (2.13 Å)
Cite:Type II Kinase Inhibitors Targeting Cys-Gatekeeper Kinases Display Orthogonality with Wild Type and Ala/Gly-Gatekeeper Kinases.
ACS Chem. Biol., 13, 2018

222415

数据于2024-07-10公开中

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