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PDB: 1 results
9MRE
From DNA-Encoded Library Screening to AM-9747 - an MTA-Cooperative PRMT5 Inhibitor with Potent Oral in vivo Efficacy
Descriptor:
2-amino-3-methyl-N-[(1R)-1-(pyrimidin-2-yl)ethyl]-N-{[5-(trifluoromethyl)pyridin-2-yl]methyl}quinoline-6-carboxamide, 5'-DEOXY-5'-METHYLTHIOADENOSINE, DI(HYDROXYETHYL)ETHER, ...
Authors:
GhimireRijal, S
,
Mukund, S.
Deposit date:
2025-01-07
Release date:
2025-03-26
Last modified:
2025-04-02
Method:
X-RAY DIFFRACTION (2.25 Å)
Cite:
From DNA-Encoded Library Screening to AM-9747 : An MTA-Cooperative PRMT5 Inhibitor with Potent Oral In Vivo Efficacy.
J.Med.Chem., 68, 2025
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数据于2025-07-23公开中