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PDB: 1 results

3MPM
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BU of 3mpm by Molmil
LCK complexed with a pyrazolopyrimidine
Descriptor: 1,2-ETHANEDIOL, 4-{(6R,7R)-7-amino-3-[3-(4-methylpiperazin-1-yl)phenyl]-6,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl}phenol, Tyrosine-protein kinase Lck
Authors:Cowan-Jacob, S.W, Rummel, G.
Deposit date:2010-04-27
Release date:2010-06-02
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:New pyrazolo[1,5a]pyrimidines as orally active inhibitors of Lck.
Bioorg.Med.Chem.Lett., 20, 2010

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数据于2024-07-17公开中

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