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PDB: 1 results
8UV0
Discovery of (4-Pyrazolyl)-2-Aminopyrimidines as Potent and Selective Inhibitors of Cyclin-Dependent Kinase 2
Descriptor:
1-{(4M)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1H-pyrazol-1-yl}-2-methylpropan-2-ol, Cyclin-dependent kinase 2
Authors:
Deller, M.C
,
Epling, L.B.
Deposit date:
2023-11-02
Release date:
2024-02-14
Last modified:
2024-03-06
Method:
X-RAY DIFFRACTION (1.55 Å)
Cite:
Discovery of (4-Pyrazolyl)-2-aminopyrimidines as Potent and Selective Inhibitors of Cyclin-Dependent Kinase 2.
J.Med.Chem., 67, 2024
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건을2024-07-17부터공개중