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PDB: 7 results
5MGG
Crystal Structure of BAZ2B bromodomain in complex with 4-chloropyridine derivative 3
Descriptor:
4-chloranyl-~{N}-methyl-pyridine-2-carboxamide, Bromodomain adjacent to zinc finger domain protein 2B
Authors:
Lolli, G
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-11-21
Release date:
2017-04-12
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (2.1 Å)
Cite:
Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
5MGJ
Crystal Structure of BAZ2A bromodomain in complex with 1-methylpyridine derivative 1
Descriptor:
Bromodomain adjacent to zinc finger domain protein 2A, ethyl 4-chloranyl-1-methyl-6-oxidanylidene-pyridine-3-carboxylate
Authors:
Lolli, G
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-11-21
Release date:
2017-04-12
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (2.1 Å)
Cite:
Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
5MGL
Crystal Structure of BAZ2A bromodomain in complex with 4-chloropyridine derivative 3
Descriptor:
4-chloranyl-~{N}-methyl-pyridine-2-carboxamide, Bromodomain adjacent to zinc finger domain protein 2A
Authors:
Lolli, G
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-11-21
Release date:
2017-04-12
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (2.651 Å)
Cite:
Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
5MGF
Crystal Structure of BAZ2B bromodomain in complex with 4-propionyl-pyrrole derivative 2
Descriptor:
Bromodomain adjacent to zinc finger domain protein 2B, methyl 4-propanoyl-1~{H}-pyrrole-2-carboxylate
Authors:
Lolli, G
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-11-21
Release date:
2017-04-12
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (1.9 Å)
Cite:
Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
5MGE
Crystal structure of BAZ2B bromodomain in complex with 1-methylpyridine derivative 1
Descriptor:
Bromodomain adjacent to zinc finger domain protein 2B, ethyl 4-chloranyl-1-methyl-6-oxidanylidene-pyridine-3-carboxylate
Authors:
Lolli, G
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-11-21
Release date:
2017-04-12
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (1.95 Å)
Cite:
Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
5MGM
Crystal Structure of BAZ2A bromodomain in complex with acetophenone derivative 4
Descriptor:
1-(3-pyrimidin-2-yloxyphenyl)ethanone, Bromodomain adjacent to zinc finger domain protein 2A
Authors:
Lolli, G
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-11-21
Release date:
2017-04-12
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (2.8 Å)
Cite:
Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
5MGK
Crystal Structure of BAZ2A bromodomain in complex with 4-propionyl-pyrrole derivative 2
Descriptor:
Bromodomain adjacent to zinc finger domain protein 2A, methyl 4-propanoyl-1~{H}-pyrrole-2-carboxylate
Authors:
Lolli, G
,
Spiliotopoulos, D
,
Caflisch, A.
Deposit date:
2016-11-21
Release date:
2017-04-12
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (2.301 Å)
Cite:
Discovery of BAZ2A bromodomain ligands.
Eur J Med Chem, 139, 2017
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건을2024-07-10부터공개중