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PDB: 1 results

9G7H
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BU of 9g7h by Molmil
Human Sirt6 in complex with ADP-ribose and the inhibitor 2-Pr
Descriptor: 2,4-bis(oxidanylidene)-1-[2-oxidanylidene-2-[[(2S)-3-oxidanylidene-3-(propylamino)-2-[3-(3-pyridin-3-yl-1,2,4-oxadiazol-5-yl)propanoylamino]propyl]amino]ethyl]pyrimidine-5-carboxamide, NAD-dependent protein deacetylase sirtuin-6, SULFATE ION, ...
Authors:You, W, Steegborn, C.
Deposit date:2024-07-21
Release date:2024-08-14
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Elucidating the Unconventional Binding Mode of a DNA-Encoded Library Hit Provides a Blueprint for Sirtuin 6 Inhibitor Development.
Chemmedchem, 2024

224931

건을2024-09-11부터공개중

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