2WMU
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![BU of 2wmu by Molmil](/molmil-images/mine/2wmu) | Crystal structure of checkpoint kinase 1 (Chk1) in complex with inhibitors | 分子名称: | 6-MORPHOLIN-4-YL-9H-PURINE, SERINE/THREONINE-PROTEIN KINASE CHK1 | 著者 | Matthews, T.P, Klair, S, Burns, S, Boxall, K, Cherry, M, Fisher, M, Westwood, I.M, Walton, M.I, McHardy, T, Cheung, K.-M.J, Van Montfort, R, Williams, D, Aherne, G.W, Garrett, M.D, Reader, J, Collins, I. | 登録日 | 2009-07-03 | 公開日 | 2009-07-28 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Identification of Inhibitors of Checkpoint Kinase 1 Through Template Screening. J.Med.Chem., 52, 2009
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1YXA
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![BU of 1yxa by Molmil](/molmil-images/mine/1yxa) | Serpina3n, a murine orthologue of human antichymotrypsin | 分子名称: | serine (or cysteine) proteinase inhibitor, clade A, member 3N | 著者 | Horvath, A.J, Irving, J.A, Law, R.H, Rossjohn, J, Bottomley, S.P, Quinsey, N.S, Pike, R.N, Coughlin, P.B, Whisstock, J.C. | 登録日 | 2005-02-20 | 公開日 | 2005-09-06 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The murine orthologue of human antichymotrypsin: a structural paradigm for clade A3 serpins. J.Biol.Chem., 280, 2005
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1L2E
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![BU of 1l2e by Molmil](/molmil-images/mine/1l2e) | Human Kallikrein 6 (hK6) Active Form with benzamidine inhibitor | 分子名称: | BENZAMIDINE, Kallikrein 6, MAGNESIUM ION | 著者 | Bernett, M.J, Blaber, S.I, Scarisbrick, I.A, Blaber, M. | 登録日 | 2002-02-20 | 公開日 | 2002-05-08 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Crystal structure and biochemical characterization of human kallikrein 6 reveals that a trypsin-like kallikrein is expressed in the central nervous system. J.Biol.Chem., 277, 2002
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2CE2
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![BU of 2ce2 by Molmil](/molmil-images/mine/2ce2) | CRYSTAL STRUCTURE ANALYSIS OF A FLUORESCENT FORM OF H-RAS P21 IN COMPLEX WITH GDP | 分子名称: | GTPASE HRAS, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Klink, B.U, Goody, R.S, Scheidig, A.J. | 登録日 | 2006-02-02 | 公開日 | 2006-08-23 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (1 Å) | 主引用文献 | A Newly Designed Microspectrofluorometer for Kinetic Studies on Protein Crystals in Combination with X-Ray Diffraction Biophys.J., 91, 2006
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1YXV
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![BU of 1yxv by Molmil](/molmil-images/mine/1yxv) | Crystal Structure of Kinase Pim1 in complex with 3,4-Dihydroxy-1-methylquinolin-2(1H)-one | 分子名称: | 3,4-DIHYDROXY-1-METHYLQUINOLIN-2(1H)-ONE, IMIDAZOLE, Proto-oncogene serine/threonine-protein kinase Pim-1 | 著者 | Kumar, A, Mandiyan, V, Suzuki, Y, Zhang, C, Rice, J, Tsai, J, Artis, D.R, Ibrahim, P, Bremer, R. | 登録日 | 2005-02-22 | 公開日 | 2005-04-26 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal Structures of Proto-oncogene Kinase Pim1: A Target of Aberrant Somatic Hypermutations in Diffuse Large Cell Lymphoma. J.Mol.Biol., 348, 2005
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2WTC
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![BU of 2wtc by Molmil](/molmil-images/mine/2wtc) | CRYSTAL STRUCTURE OF CHK2 IN COMPLEX WITH AN INHIBITOR | 分子名称: | 4-[2-AMINO-5-(4-HYDROXY-3-METHOXYPHENYL)PYRIDIN-3-YL]BENZAMIDE, NITRATE ION, SERINE/THREONINE-PROTEIN KINASE CHK2 | 著者 | Hilton, S, Naud, S, Caldwell, J.J, Boxall, K, Burns, S, Anderson, V.E, Antoni, L, Allen, C.E, Pearl, L.H, Oliver, A.W, Aherne, G.W, Garrett, M.D, Collins, I. | 登録日 | 2009-09-15 | 公開日 | 2009-12-29 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Identification and Characterisation of 2-Aminopyridine Inhibitors of Checkpoint Kinase 2 Bioorg.Med.Chem., 18, 2010
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1YWP
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![BU of 1ywp by Molmil](/molmil-images/mine/1ywp) | Phospholipase Cgamma1 SH3 | 分子名称: | 1-phosphatidylinositol-4,5-bisphosphate phosphodiesterase gamma 1 | 著者 | Deng, L, Velikovsky, C.A, Swaminathan, C.P, Cho, S, Mariuzza, R.A. | 登録日 | 2005-02-18 | 公開日 | 2005-08-16 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structural Basis for Recognition of the T Cell Adaptor Protein SLP-76 by the SH3 Domain of Phospholipase Cgamma1 J.Mol.Biol., 352, 2005
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1YWV
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![BU of 1ywv by Molmil](/molmil-images/mine/1ywv) | Crystal Structures of Proto-Oncogene Kinase Pim1: a Target of Aberrant Somatic Hypermutations in Diffuse Large Cell Lymphoma | 分子名称: | IMIDAZOLE, Proto-oncogene serine/threonine-protein kinase Pim-1 | 著者 | Kumar, A, Mandiyan, V, Suzuki, Y, Zhang, C, Rice, J, Tsai, J, Artis, D.R, Ibrahim, P, Bremer, R. | 登録日 | 2005-02-18 | 公開日 | 2005-04-26 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structures of proto-oncogene kinase Pim1: a target of aberrant somatic hypermutations in diffuse large cell lymphoma. J.Mol.Biol., 348, 2005
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1LJJ
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1TNG
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![BU of 1tng by Molmil](/molmil-images/mine/1tng) | |
1LJW
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![BU of 1ljw by Molmil](/molmil-images/mine/1ljw) | Crystal Structure of Human Carbonmonoxy Hemoglobin at 2.16 A: A Snapshot of the Allosteric Transition | 分子名称: | CARBON MONOXIDE, PHOSPHATE ION, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Safo, M.K, Burnett, J.C, Musayev, F.N, Nokuri, S, Abraham, D.J. | 登録日 | 2002-04-22 | 公開日 | 2002-05-01 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.16 Å) | 主引用文献 | Structure of human carbonmonoxyhemoglobin at 2.16 A: a snapshot of the allosteric transition. Acta Crystallogr.,Sect.D, 58, 2002
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2CPN
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![BU of 2cpn by Molmil](/molmil-images/mine/2cpn) | Solution structure of the second dsRBD of TAR RNA-binding protein 2 | 分子名称: | TAR RNA-binding protein 2 | 著者 | Nagata, T, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-19 | 公開日 | 2005-11-19 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the second dsRBD of TAR RNA-binding protein 2 To be Published
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2CPD
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![BU of 2cpd by Molmil](/molmil-images/mine/2cpd) | Solution structure of the RNA recognition motif of human APOBEC-1 complementation factor, ACF | 分子名称: | APOBEC-1 stimulating protein | 著者 | Nagata, T, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-19 | 公開日 | 2005-11-19 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the RNA recognition motif of human APOBEC-1 complementation factor, ACF To be Published
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2CPX
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![BU of 2cpx by Molmil](/molmil-images/mine/2cpx) | solution structure of RNA binding domain in Hypothetical protein FLJ11016 | 分子名称: | Hypothetical protein FLJ11016 | 著者 | Tsuda, K, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-19 | 公開日 | 2005-11-19 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | solution structure of RNA binding domain in Hypothetical protein FLJ11016 To be Published
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1TRM
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2CQH
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![BU of 2cqh by Molmil](/molmil-images/mine/2cqh) | Solution structure of the RNA binding domain of IGF-II mRNA-binding protein 2 | 分子名称: | IGF-II mRNA-binding protein 2 isoform a | 著者 | Suzuki, S, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-20 | 公開日 | 2005-11-20 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the RNA binding domain of IGF-II mRNA-binding protein 2 To be Published
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2CQX
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![BU of 2cqx by Molmil](/molmil-images/mine/2cqx) | Solution structure of RSGI RUH-034, a homeodomain from mouse cDNA | 分子名称: | LAG1 longevity assurance homolog 5 | 著者 | Ruhul Momen, A.Z.M, Onuki, H, Hirota, H, Tomizawa, T, Koshiba, S, Kigawa, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-20 | 公開日 | 2005-11-20 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of RSGI RUH-034, a homeodomain from mouse cDNA To be Published
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1YZL
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![BU of 1yzl by Molmil](/molmil-images/mine/1yzl) | GppNHp-Bound Rab9 GTPase | 分子名称: | MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-GUANYLATE ESTER, Ras-related protein Rab-9A | 著者 | Eathiraj, S, Pan, X, Ritacco, C, Lambright, D.G. | 登録日 | 2005-02-28 | 公開日 | 2005-07-26 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structural basis of family-wide Rab GTPase recognition by rabenosyn-5. Nature, 436, 2005
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2CRH
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1Z0I
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![BU of 1z0i by Molmil](/molmil-images/mine/1z0i) | GDP-Bound Rab21 GTPase | 分子名称: | GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Ras-related protein Rab-21 | 著者 | Eathiraj, S, Pan, X, Ritacco, C, Lambright, D.G. | 登録日 | 2005-03-01 | 公開日 | 2005-07-26 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | Structural basis of family-wide Rab GTPase recognition by rabenosyn-5. Nature, 436, 2005
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1V2N
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![BU of 1v2n by Molmil](/molmil-images/mine/1v2n) | Potent factor XA inhibitor in complex with bovine trypsin variant X(99/175/190)bT | 分子名称: | 2,7-BIS-(4-AMIDINOBENZYLIDENE)-CYCLOHEPTAN-1-ONE, CALCIUM ION, Trypsin | 著者 | Rauh, D, Klebe, G, Stubbs, M.T. | 登録日 | 2003-10-17 | 公開日 | 2004-06-01 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Understanding protein-ligand interactions: the price of protein flexibility J.Mol.Biol., 335, 2004
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1Z1R
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![BU of 1z1r by Molmil](/molmil-images/mine/1z1r) | HIV-1 protease complexed with Macrocyclic peptidomimetic inhibitor 2 | 分子名称: | 2-[(8S,11S)-11-{(1R)-1-HYDROXY-2-[ISOPENTYL(PHENYLSULFONYL)AMINO]ETHYL}-6,9-DIOXO-2-OXA-7,10-DIAZABICYCLO[11.2.2]HEPTADECA-1(15),13,16-TRIEN-8-YL]ACETAMIDE, Pol polyprotein, SULFATE ION | 著者 | Martin, J.L, Begun, J, Schindeler, A, Wickramasinghe, W.A, Alewood, D, Alewood, P.F, Bergman, D.A, Brinkworth, R.I, Abbenante, G, March, D.R, Reid, R.C, Fairlie, D.P. | 登録日 | 2005-03-06 | 公開日 | 2005-03-22 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease Biochemistry, 38, 1999
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2CUF
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![BU of 2cuf by Molmil](/molmil-images/mine/2cuf) | Solution structure of the homeobox domain of the human hypothetical protein FLJ21616 | 分子名称: | FLJ21616 protein | 著者 | Ohnishi, S, Kigawa, T, Tomizawa, T, Koshiba, S, Inoue, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-05-26 | 公開日 | 2005-11-26 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the homeobox domain of the human hypothetical protein FLJ21616 To be Published
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1KZA
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![BU of 1kza by Molmil](/molmil-images/mine/1kza) | Complex of MBP-C and Man-a13-Man | 分子名称: | CALCIUM ION, CHLORIDE ION, MANNOSE-BINDING PROTEIN C, ... | 著者 | Ng, K.K, Kolatkar, A.R, Park-Snyder, S, Feinberg, H, Clark, D.A, Drickamer, K, Weis, W.I. | 登録日 | 2002-02-06 | 公開日 | 2002-07-05 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Orientation of bound ligands in mannose-binding proteins. Implications for multivalent ligand recognition. J.Biol.Chem., 277, 2002
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2WQN
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![BU of 2wqn by Molmil](/molmil-images/mine/2wqn) | Structure of ADP-bound human Nek7 | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, NICKEL (II) ION, ... | 著者 | Richards, M.W, Bayliss, R. | 登録日 | 2009-08-24 | 公開日 | 2009-12-08 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | An Autoinhibitory Tyrosine Motif in the Cell-Cycle- Regulated Nek7 Kinase is Released Through Binding of Nek9. Mol.Cell, 36, 2009
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