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7E62
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BU of 7e62 by Molmil
Mouse TAB2 NZF in complex with Lys6-linked diubiquitin
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, TGF-beta-activated kinase 1 and MAP3K7-binding protein 2, Ubiquitin, ...
著者Sato, Y, Li, Y, Okatsu, K, Fukai, S.
登録日2021-02-21
公開日2021-08-18
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献Structural basis for specific recognition of K6-linked polyubiquitin chains by the TAB2 NZF domain.
Biophys.J., 120, 2021
1T9Z
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BU of 1t9z by Molmil
Three-dimensional structure of a RNA-polymerase II binding protein.
分子名称: CITRIC ACID, Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1, MAGNESIUM ION
著者Kamenski, T, Heilmeier, S, Meinhart, A, Cramer, P.
登録日2004-05-19
公開日2004-08-31
最終更新日2021-10-27
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structure and Mechanism of RNA Polymerase II CTD Phosphatases.
Mol.Cell, 15, 2004
4EEP
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BU of 4eep by Molmil
Crystal structure of LOV2 domain of Arabidopsis thaliana phototropin 2
分子名称: FLAVIN MONONUCLEOTIDE, Phototropin-2
著者Hitomi, K, Christie, J.M, Arvai, A.S, Hartfield, K.A, Pratt, A.J, Tainer, J.A, Getzoff, E.D.
登録日2012-03-28
公開日2012-05-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural Tuning of the Fluorescent Protein iLOV for Improved Photostability.
J.Biol.Chem., 287, 2012
4EH8
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BU of 4eh8 by Molmil
Human p38 MAP kinase in complex with NP-F7 and RL87
分子名称: Mitogen-activated protein kinase 14, N~4~-cyclopropyl-2-phenylquinazoline-4,7-diamine, [3-(benzyloxy)phenyl]methanol
著者Over, B, Gruetter, C, Waldmann, H, Rauh, D.
登録日2012-04-02
公開日2012-12-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Natural-product-derived fragments for fragment-based ligand discovery.
Nat Chem, 5, 2012
2Q2Y
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BU of 2q2y by Molmil
Crystal Structure of KSP in complex with Inhibitor 1
分子名称: 1-{(3R,3AR)-3-[3-(4-ACETYLPIPERAZIN-1-YL)PROPYL]-8-FLUORO-3-PHENYL-3A,4-DIHYDRO-3H-PYRAZOLO[5,1-C][1,4]BENZOXAZIN-2-YL}ETHANONE, ADENOSINE-5'-DIPHOSPHATE, Kinesin-like protein KIF11, ...
著者Yan, Y.
登録日2007-05-29
公開日2007-09-18
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Kinesin spindle protein (KSP) inhibitors. Part 8: Design and synthesis of 1,4-diaryl-4,5-dihydropyrazoles as potent inhibitors of the mitotic kinesin KSP.
Bioorg.Med.Chem.Lett., 17, 2007
1TA0
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BU of 1ta0 by Molmil
Three-dimensional structure of a RNA-polymerase II binding protein with associated ligand.
分子名称: CITRIC ACID, Carboxy-terminal domain RNA polymerase II polypeptide A small phosphatase 1, MAGNESIUM ION
著者Kamenski, T, Heilmeier, S, Meinhart, T, Cramer, P.
登録日2004-05-19
公開日2004-08-31
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure and Mechanism of RNA Polymerase II CTD Phosphatases.
Mol.Cell, 15, 2004
2N7D
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BU of 2n7d by Molmil
Solution structure of the UBL domain of human Ddi2
分子名称: Protein DDI1 homolog 2
著者Siva, M, Grantz Saskova, K, Veverka, V.
登録日2015-09-08
公開日2016-07-20
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Human DNA-Damage-Inducible 2 Protein Is Structurally and Functionally Distinct from Its Yeast Ortholog.
Sci Rep, 6, 2016
4BU7
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BU of 4bu7 by Molmil
Crystal structure of human tankyrase 2 in complex with 2-(4- bromophenyl)-3,4-dihydroquinazolin-4-one
分子名称: 2-(4-bromophenyl)-3,4-dihydroquinazolin-4-one, GLYCEROL, SULFATE ION, ...
著者Haikarainen, T, Narwal, M, Lehtio, L.
登録日2013-06-20
公開日2013-10-30
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Para-Substituted 2-Phenyl-3,4-Dihydroquinazolin-4-Ones as Potent and Selective Tankyrase Inhibitors.
Chemmedchem, 8, 2013
2NZ7
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BU of 2nz7 by Molmil
Crystal Structure Analysis of Caspase-recruitment Domain (CARD) of Nod1
分子名称: Caspase recruitment domain-containing protein 4
著者Thiagarajan, S, Robbins, S.L, Dubas, R.L, Park, Y.C.
登録日2006-11-22
公開日2007-12-04
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Monomer/dimer transition of the caspase-recruitment domain of human Nod1
Biochemistry, 47, 2008
4EH4
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BU of 4eh4 by Molmil
Human p38 MAP kinase in complex with NP-F3 and RL87
分子名称: Mitogen-activated protein kinase 14, N~4~-cyclopropyl-2-phenylquinazoline-4,7-diamine, phenyl(piperidin-1-yl)methanone
著者Over, B, Gruetter, C, Waldmann, H, Rauh, D.
登録日2012-04-02
公開日2012-12-05
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Natural-product-derived fragments for fragment-based ligand discovery.
Nat Chem, 5, 2012
7FSV
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BU of 7fsv by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1454310449
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSR
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BU of 7fsr by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z54615640
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT9
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BU of 7ft9 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z45636695
分子名称: 1,2-ETHANEDIOL, 4-[(METHYLSULFONYL)AMINO]BENZOIC ACID, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.77 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FTA
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BU of 7fta by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z228589380
分子名称: 1,2-ETHANEDIOL, 3-[(pyrimidin-2-yl)amino]benzoic acid, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSJ
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BU of 7fsj by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z57744712
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSU
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BU of 7fsu by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z729726784
分子名称: 1,2-ETHANEDIOL, 2-cyclopentyl-N-(3-methyl-1,2,4-oxadiazol-5-yl)acetamide, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FTB
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BU of 7ftb by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1198269757
分子名称: 1,2-ETHANEDIOL, D-GLUTAMIC ACID, GLYCINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FST
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BU of 7fst by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z26968795
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSM
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BU of 7fsm by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z763030030
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSP
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BU of 7fsp by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1650168321
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.86 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSG
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BU of 7fsg by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z56772132
分子名称: (5R)-5-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione, 1,2-ETHANEDIOL, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSW
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BU of 7fsw by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z169675004
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSY
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BU of 7fsy by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1148165337
分子名称: 1,2-ETHANEDIOL, 2-(1H-indazol-1-yl)-N,N-dimethylacetamide, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT7
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BU of 7ft7 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z57127349
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.78 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT2
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BU of 7ft2 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z235449082
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.04 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published

222415

件を2024-07-10に公開中

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