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8JTB
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BU of 8jtb by Molmil
VMAT2 complex with dopamine
分子名称: L-DOPAMINE, Synaptic vesicular amine transporter
著者Jiang, D.H, Wu, D.
登録日2023-06-21
公開日2024-05-08
実験手法ELECTRON MICROSCOPY (2.93 Å)
主引用文献VMAT2 complex with dopamine
To Be Published
8OMU
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BU of 8omu by Molmil
Cryo-EM structure of rat SLC22A6 bound to alpha-ketoglutaric acid in a low occupancy state
分子名称: Solute carrier family 22 member 6, Synthetic nanobody (Sybody)
著者Parker, J.L, Kato, T, Newstead, S.
登録日2023-03-31
公開日2023-07-19
最終更新日2023-11-22
実験手法ELECTRON MICROSCOPY (3.43 Å)
主引用文献Molecular basis for selective uptake and elimination of organic anions in the kidney by OAT1.
Nat.Struct.Mol.Biol., 30, 2023
8JTC
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BU of 8jtc by Molmil
Human VMAT2 complex with reserpine
分子名称: Synaptic vesicular amine transporter, reserpine
著者Jiang, D.H, Wu, D.
登録日2023-06-21
公開日2023-11-29
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (3.52 Å)
主引用文献Transport and inhibition mechanisms of human VMAT2.
Nature, 626, 2024
8JTA
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BU of 8jta by Molmil
Human VMAT2 complex with tetrabenazine
分子名称: Synaptic vesicular amine transporter, tetrabenazine
著者Jiang, D.H, Wu, D.
登録日2023-06-21
公開日2023-11-29
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (3.36 Å)
主引用文献Transport and inhibition mechanisms of human VMAT2.
Nature, 626, 2024
8JSW
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BU of 8jsw by Molmil
Human VMAT2 complex with serotonin
分子名称: SEROTONIN, Synaptic vesicular amine transporter
著者Jiang, D.H, Wu, D.
登録日2023-06-20
公開日2023-11-29
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (2.84 Å)
主引用文献Transport and inhibition mechanisms of human VMAT2.
Nature, 626, 2024
8JT9
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BU of 8jt9 by Molmil
Human VMAT2 complex with ketanserin
分子名称: 3-[2-[4-(4-fluorophenyl)carbonylpiperidin-1-yl]ethyl]-1~{H}-quinazoline-2,4-dione, Synaptic vesicular amine transporter
著者Jiang, D.H, Wu, D.
登録日2023-06-21
公開日2023-11-29
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (2.97 Å)
主引用文献Transport and inhibition mechanisms of human VMAT2.
Nature, 626, 2024
8PNL
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BU of 8pnl by Molmil
Outward-open conformation of a Major Facilitator Superfamily (MFS) transporter MHAS2168, a homologue of Rv1410 from M. tuberculosis, in complex with an alpaca nanobody
分子名称: Nb_H2, Putative triacylglyceride transporter
著者Remm, S, Schoeppe, J, Hutter, C.A.J, Gonda, I, Seeger, M.A.
登録日2023-06-30
公開日2023-10-18
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural basis for triacylglyceride extraction from mycobacterial inner membrane by MFS transporter Rv1410.
Nat Commun, 14, 2023
8KAE
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BU of 8kae by Molmil
16d-bound human SPNS2
分子名称: 3-[3-(4-decylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-amine, NbFab chain L, NbFab-H chain, ...
著者He, Y, Duan, Y.
登録日2023-08-03
公開日2024-01-03
最終更新日2024-02-21
実験手法ELECTRON MICROSCOPY (3.18 Å)
主引用文献Structural basis of Sphingosine-1-phosphate transport via human SPNS2.
Cell Res., 34, 2024
8UO8
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BU of 8uo8 by Molmil
Structure of synaptic vesicle protein 2B with padsevonil
分子名称: (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, (4R)-4-(2-chloro-2,2-difluoroethyl)-1-{[(4R)-2-(methoxymethyl)-6-(trifluoromethyl)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]methyl}pyrrolidin-2-one, 1,2-DIDECANOYL-SN-GLYCERO-3-[PHOSPHO-L-SERINE], ...
著者Martin, M.F, Mittal, A, Levin, E, Adams, C, Yang, M, Ledecq, M, Horyani, P.S, Coleman, J.A.
登録日2023-10-19
公開日2024-05-22
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Structure of synaptic vesicle protein 2B with padsevonil
To Be Published
8JHQ
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BU of 8jhq by Molmil
Cryo-EM structure of human S1P transporter SPNS2 bound with S1P
分子名称: (2S,3R,4E)-2-amino-3-hydroxyoctadec-4-en-1-yl dihydrogen phosphate, Sphingosine-1-phosphate transporter SPNS2,GlgA glycogen synthase
著者Pang, B, Yu, L.Y, Ren, R.B.
登録日2023-05-25
公開日2024-01-10
最終更新日2024-02-14
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Molecular basis of Spns2-facilitated sphingosine-1-phosphate transport.
Cell Res., 34, 2024
8JLF
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BU of 8jlf by Molmil
Cryo-EM structure of SV2A in complex with BoNT/A2 Hc
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, Botulinum neurotoxin, ...
著者Yamagata, A.
登録日2023-06-02
公開日2024-05-01
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.01 Å)
主引用文献Structural basis for antiepileptic drugs and botulinum neurotoxin recognition of SV2A.
Nat Commun, 15, 2024
8JLC
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BU of 8jlc by Molmil
Cryo-EM structure of SV2A in complex with BoNT/A2 Hc and levetiracetam
分子名称: (2S)-2-(2-oxidanylidenepyrrolidin-1-yl)butanamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Yamagata, A.
登録日2023-06-02
公開日2024-05-01
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (2.88 Å)
主引用文献Structural basis for antiepileptic drugs and botulinum neurotoxin recognition of SV2A.
Nat Commun, 15, 2024
8JS8
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BU of 8js8 by Molmil
Cryo-EM structure of SV2A in complex with BoNT/A2 Hc and levetiracetam
分子名称: (2S)-2-(2-oxidanylidenepyrrolidin-1-yl)butanamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Yamagata, A.
登録日2023-06-19
公開日2024-05-01
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (2.88 Å)
主引用文献Structural basis for antiepileptic drugs and botulinum neurotoxin recognition of SV2A.
Nat Commun, 15, 2024
8JS9
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BU of 8js9 by Molmil
Cryo-EM structure of SV2A in complex with BoNT/A2 Hc
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, Botulinum neurotoxin, ...
著者Yamagata, A.
登録日2023-06-19
公開日2024-05-01
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.01 Å)
主引用文献Structural basis for antiepileptic drugs and botulinum neurotoxin recognition of SV2A.
Nat Commun, 15, 2024
8JLH
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BU of 8jlh by Molmil
Cryo-EM structure of SV2A dimer in complex with BoNT/A2 Hc and levetiracetam
分子名称: (2S)-2-(2-oxidanylidenepyrrolidin-1-yl)butanamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Yamagata, A.
登録日2023-06-02
公開日2024-05-01
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Structural basis for antiepileptic drugs and botulinum neurotoxin recognition of SV2A.
Nat Commun, 15, 2024
8K77
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BU of 8k77 by Molmil
Cryo-EM structure of SV2A in complex with BoNT/A2 Hc and brivaracetam
分子名称: (2S)-2-[(4R)-2-oxidanylidene-4-propyl-pyrrolidin-1-yl]butanamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Yamagata, A.
登録日2023-07-26
公開日2024-05-01
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (3.11 Å)
主引用文献Structural basis for antiepileptic drugs and botulinum neurotoxin recognition of SV2A.
Nat Commun, 15, 2024

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件を2024-06-12に公開中

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