4UZ0
| Crystal Structure of apoptosis repressor with CARD (ARC) | 分子名称: | GLYCEROL, NUCLEOLAR PROTEIN 3 | 著者 | Kim, S.H, Jeong, J.H, Jang, T.H, Kim, Y.G, Park, H.H. | 登録日 | 2014-09-04 | 公開日 | 2015-07-01 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (2.399 Å) | 主引用文献 | Crystal Structure of Caspase Recruiting Domain (Card) of Apoptosis Repressor with Card (Arc) and its Implication in Inhibition of Apoptosis. Sci.Rep., 5, 2015
|
|
4UU9
| Crystal structure of the human c5a in complex with MEDI7814 a neutralising antibody | 分子名称: | COMPLEMENT C5, MEDI7814, SULFATE ION | 著者 | Colley, C, Sridharan, S, Dobson, C, Popovic, B, Debreczeni, J.E, Hargreaves, D, Edwards, B, Brennan, J, England, L, Fung, S, An Eghobamien, L, Sivars, U, Woods, R, Flavell, L, Renshaw, G.J, Wickson, K, Wilkinson, T, Davies, R, Bonnell, J, Warrener, P, Howes, R, Vaughan, T. | 登録日 | 2014-07-25 | 公開日 | 2015-08-12 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (2.12 Å) | 主引用文献 | Structure and characterization of a high affinity C5a monoclonal antibody that blocks binding to C5aR1 and C5aR2 receptors. MAbs, 10, 2018
|
|
8H45
| Blasnase-T13A/P55N | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
|
|
2UUY
| Structure of a tick tryptase inhibitor in complex with bovine trypsin | 分子名称: | CALCIUM ION, CATIONIC TRYPSIN, CHLORIDE ION, ... | 著者 | Siebold, C, Paesen, G.C, Harlos, K, Peacey, M.F, Nuttall, P.A, Stuart, D.I. | 登録日 | 2007-03-08 | 公開日 | 2007-04-10 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | A Tick Protein with a Modified Kunitz Fold Inhibits Human Tryptase. J.Mol.Biol., 368, 2007
|
|
2UVH
| |
4UYK
| Crystal structure of a Signal Recognition Particle Alu domain in the elongation arrest conformation | 分子名称: | SIGNAL RECOGNITION PARTICLE 14 KDA PROTEIN, SIGNAL RECOGNITION PARTICLE 9 KDA PROTEIN, SRP RNA | 著者 | Bousset, L, Mary, C, Brooks, M.A, Scherrer, A, Strub, K, Cusack, S. | 登録日 | 2014-09-01 | 公開日 | 2014-11-05 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (3.22 Å) | 主引用文献 | Crystal Structure of a Signal Recognition Particle Alu Domain in the Elongation Arrest Conformation. RNA, 20, 2014
|
|
8H48
| Blasnase-T13A/P55F with L-asn | 分子名称: | ASPARAGINE, FORMIC ACID, L-asparaginase, ... | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
|
|
2UVK
| |
8H6I
| The crystal structure of SARS-CoV-2 3C-like protease Double Mutant (L50F and E166V) in complex with a traditional Chinese Medicine Inhibitors | 分子名称: | (1beta,6beta,7beta,8alpha,9beta,10alpha,13alpha,14R,16beta)-1,6,7,14-tetrahydroxy-7,20-epoxykauran-15-one, 3C-like proteinase nsp5 | 著者 | Lin, M, Liu, X. | 登録日 | 2022-10-17 | 公開日 | 2023-10-11 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Molecular mechanisms of SARS-CoV-2 resistance to nirmatrelvir. Nature, 622, 2023
|
|
4V2P
| Ketosynthase MxnB | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, CHLORIDE ION, KETOSYNTHASE, ... | 著者 | Koehnke, J. | 登録日 | 2014-10-13 | 公開日 | 2015-08-26 | 最終更新日 | 2024-10-16 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | In vitro reconstitution of alpha-pyrone ring formation in myxopyronin biosynthesis. Chem Sci, 6, 2015
|
|
2UVY
| Structure of PKA-PKB chimera complexed with methyl-(4-(9H-purin-6-yl)- benzyl)-amine | 分子名称: | CAMP-DEPENDENT PROTEIN KINASE INHIBITOR ALPHA, CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT, ... | 著者 | Davies, T.G, Donald, A, McHardy, T, Rowlands, M.G, Hunter, L.J, Boyle, R.G, Aherne, G.W, Garrett, M.D, Collins, I. | 登録日 | 2007-03-15 | 公開日 | 2007-05-08 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Rapid Evolution of 6-Phenylpurine Inhibitors of Protein Kinase B Through Structure-Based Design J.Med.Chem., 50, 2007
|
|
4V7Z
| Structure of the Thermus thermophilus 70S ribosome complexed with telithromycin. | 分子名称: | 16S rRNA, 23S ribosomal RNA, 30S ribosomal protein S10, ... | 著者 | Bulkley, D.P, Innis, C.A, Blaha, G, Steitz, T.A. | 登録日 | 2010-08-18 | 公開日 | 2014-07-09 | 最終更新日 | 2021-01-27 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Revisiting the structures of several antibiotics bound to the bacterial ribosome. Proc.Natl.Acad.Sci.USA, 107, 2010
|
|
8H7K
| |
8H4Q
| |
2UVG
| |
2UW5
| Structure of PKA-PKB chimera complexed with (R)-2-(4-chloro-phenyl)- 2-(4-1H-pyrazol-4-yl)-phenyl)-ethylamine | 分子名称: | (2R)-2-(4-CHLOROPHENYL)-2-[4-(1H-PYRAZOL-4-YL)PHENYL]ETHANAMINE, CAMP-DEPENDENT PROTEIN KINASE INHIBITOR ALPHA, CAMP-DEPENDENT PROTEIN KINASE, ... | 著者 | Davies, T.G, Saxty, G, Woodhead, S.J, Berdini, V, Verdonk, M.L, Wyatt, P.G, Boyle, R.G, Barford, D, Downham, R, Garrett, M.D, Carr, R.A. | 登録日 | 2007-03-19 | 公開日 | 2007-05-08 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (2.14 Å) | 主引用文献 | Identification of Inhibitors of Protein Kinase B Using Fragment-Based Lead Discovery J.Med.Chem., 50, 2007
|
|
8H5K
| |
4V8X
| Structure of Thermus thermophilus ribosome | 分子名称: | 16S ribosomal RNA, 23S ribosomal RNA, 30S RIBOSOMAL PROTEIN S10, ... | 著者 | Feng, S, Chen, Y, Kamada, K, Wang, H, Tang, K, Wang, M, Gao, Y.G. | 登録日 | 2013-07-19 | 公開日 | 2014-07-09 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.35 Å) | 主引用文献 | Yoeb-Ribosome Structure: A Canonical Rnase that Requires the Ribosome for its Specific Activity. Nucleic Acids Res., 41, 2013
|
|
2UUI
| Crystal structure of Human Leukotriene C4 Synthase | 分子名称: | DODECYL-BETA-D-MALTOSIDE, LEUKOTRIENE C4 SYNTHASE, NICKEL (II) ION, ... | 著者 | Martinez Molina, D, Wetterholm, A, Kohl, A, McCarthy, A.A, Niegowski, D, Ohlson, E, Hammarberg, T, Eshaghi, S, Haeggstrom, J.Z, Nordlund, P. | 登録日 | 2007-03-02 | 公開日 | 2007-07-17 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural Basis for Synthesis of Inflammatory Mediators by Human Leukotriene C4 Synthase. Nature, 448, 2007
|
|
8H49
| Blasnase-M57P | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
|
|
4V66
| Structure of the E. coli ribosome and the tRNAs in Post-accommodation state | 分子名称: | 16S rRNA, 23S rRNA, 30S ribosomal protein S10, ... | 著者 | Devkota, B, Caulfield, T.R, Tan, R.-Z, Harvey, S.C. | 登録日 | 2008-08-03 | 公開日 | 2014-07-09 | 最終更新日 | 2024-02-28 | 実験手法 | ELECTRON MICROSCOPY (9 Å) | 主引用文献 | The Structure of the E. coli Ribosome Before and After Accommodation: Implications for Proofreading To be Published
|
|
8H4A
| Blasnase-T13A/M57P | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
|
|
2UUN
| Crystal structure of C-phycocyanin from Phormidium, Lyngbya spp. (Marine) and Spirulina sp. (Fresh water) shows two different ways of energy transfer between two hexamers. | 分子名称: | BILIVERDINE IX ALPHA, C-PHYCOCYANIN, PHYCOCYANOBILIN | 著者 | Satyanarayana, L, Patel, A, Mishra, S, K Ghosh, P, Suresh, C.G. | 登録日 | 2007-03-05 | 公開日 | 2008-05-13 | 最終更新日 | 2011-07-13 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Crystal Structure of C-Phycocyanin from Phormidium, Lyngbya Spp. (Marine) and Spirulina Sp. (Fresh Water) Shows Two Different Ways of Energy Transfer between Two Hexamers. To be Published
|
|
4V6L
| Structural insights into cognate vs. near-cognate discrimination during decoding. | 分子名称: | 16S ribosomal RNA, 30S ribosomal protein S10, 30S ribosomal protein S11, ... | 著者 | Agirrezabala, X, Schreiner, E, Trabuco, L.G, Lei, J, Ortiz-Meoz, R.F, Schulten, K, Green, R, Frank, J. | 登録日 | 2011-01-07 | 公開日 | 2014-07-09 | 最終更新日 | 2024-02-28 | 実験手法 | ELECTRON MICROSCOPY (13.2 Å) | 主引用文献 | Structural insights into cognate versus near-cognate discrimination during decoding. Embo J., 30, 2011
|
|
8H4C
| Blasnase-T13A/M57P | 分子名称: | FORMIC ACID, L-asparaginase, MAGNESIUM ION | 著者 | Lu, F, Wang, W, Chi, H, Ran, T. | 登録日 | 2022-10-10 | 公開日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Structure-based rational design of Bacillus licheniformis L-asparaginase with low/no D-asparaginase activity for a safer enzyme To Be Published
|
|