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1AU9
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SUBTILISIN BPN' MUTANT 8324 IN CITRATE
分子名称: CALCIUM ION, ISOPROPYL ALCOHOL, SUBTILISIN BPN', ...
著者Whitlow, M, Howard, A.J, Wood, J.F.
登録日1997-09-12
公開日1997-12-31
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Large increases in general stability for subtilisin BPN' through incremental changes in the free energy of unfolding.
Biochemistry, 28, 1989
1DJW
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BU of 1djw by Molmil
PHOSPHOINOSITIDE-SPECIFIC PHOSPHOLIPASE C-DELTA1 FROM RAT COMPLEXED WITH INOSITOL-2-METHYLENE-1,2-CYCLIC-MONOPHOSPHONATE
分子名称: ACETATE ION, CALCIUM ION, INOSITOL-2-METHYLENE-1,2-CYCLIC-MONOPHOSPHATE, ...
著者Essen, L.-O, Perisic, O, Williams, R.L.
登録日1996-08-24
公開日1997-07-23
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Structural mapping of the catalytic mechanism for a mammalian phosphoinositide-specific phospholipase C.
Biochemistry, 36, 1997
1U3T
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Crystal Structure of Human Alcohol Dehydrogenase Alpha-Alpha Isoform Complexed with N-Cyclopentyl-N-Cyclobutylformamide Determined to 2.5 Angstrom Resolution
分子名称: Alcohol dehydrogenase alpha chain, CYCLOBUTYL(CYCLOPENTYL)FORMAMIDE, NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ...
著者Gibbons, B.J, Hurley, T.D.
登録日2004-07-23
公開日2004-10-26
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献Structure of three class I human alcohol dehydrogenases complexed with isoenzyme specific formamide inhibitors
Biochemistry, 43, 2004
1DLU
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BU of 1dlu by Molmil
UNLIGANDED BIOSYNTHETIC THIOLASE FROM ZOOGLOEA RAMIGERA
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, BIOSYNTHETIC THIOLASE, SULFATE ION
著者Modis, Y, Wierenga, R.K.
登録日1999-12-12
公開日2000-04-24
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Crystallographic analysis of the reaction pathway of Zoogloea ramigera biosynthetic thiolase.
J.Mol.Biol., 297, 2000
4GW1
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BU of 4gw1 by Molmil
cQFD Meditope
分子名称: Fab heavy chain, Fab light chain, PHOSPHATE ION, ...
著者Donaldson, J.M, Zer, C, Avery, K.N, Bzymek, K.P, Horne, D.A, Williams, J.C.
登録日2012-08-31
公開日2013-10-09
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.24 Å)
主引用文献Identification and grafting of a unique peptide-binding site in the Fab framework of monoclonal antibodies.
Proc.Natl.Acad.Sci.USA, 110, 2013
1UBN
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BU of 1ubn by Molmil
SELENOSUBTILISIN BPN
分子名称: CALCIUM ION, PROTEIN (SELENOSUBTILISIN BPN)
著者McRee, D.E, McTigue, M, Hilvert, D.
登録日1999-06-02
公開日1999-06-08
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Electric fields in active sites: substrate switching from null to strong fields in thiol- and selenol-subtilisins.
Biochemistry, 38, 1999
1DM3
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BU of 1dm3 by Molmil
ACETYLATED BIOSYNTHETIC THIOLASE FROM ZOOGLOEA RAMIGERA IN COMPLEX WITH ACETYL-COA
分子名称: ACETYL COENZYME *A, BIOSYNTHETIC THIOLASE ACETYLATED AT CYS89, SULFATE ION
著者Modis, Y, Wierenga, R.K.
登録日1999-12-13
公開日2001-08-29
最終更新日2017-10-04
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystallographic analysis of the reaction pathway of Zoogloea ramigera biosynthetic thiolase.
J.Mol.Biol., 297, 2000
1DJX
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PHOSPHOINOSITIDE-SPECIFIC PHOSPHOLIPASE C-DELTA1 FROM RAT COMPLEXED WITH INOSITOL-1,4,5-TRISPHOSPHATE
分子名称: ACETATE ION, CALCIUM ION, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, ...
著者Essen, L.-O, Perisic, O, Williams, R.L.
登録日1996-08-24
公開日1997-07-07
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural mapping of the catalytic mechanism for a mammalian phosphoinositide-specific phospholipase C.
Biochemistry, 36, 1997
1SUP
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BU of 1sup by Molmil
SUBTILISIN BPN' AT 1.6 ANGSTROMS RESOLUTION: ANALYSIS OF DISCRETE DISORDER AND COMPARISON OF CRYSTAL FORMS
分子名称: CALCIUM ION, SODIUM ION, SUBTILISIN BPN', ...
著者Gallagher, D.T, Oliver, J.D, Betzel, C, Gilliland, G.L.
登録日1995-08-14
公開日1995-11-14
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Subtilisin BPN' at 1.6 A resolution: analysis for discrete disorder and comparison of crystal forms.
Acta Crystallogr.,Sect.D, 52, 1996
4FNH
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BU of 4fnh by Molmil
Crystal structure of IsdI-W66Y in complex with heme
分子名称: Heme-degrading monooxygenase isdI, PROTOPORPHYRIN IX CONTAINING FE
著者Ukpabi, G.N, Murphy, M.E.P.
登録日2012-06-19
公開日2012-08-22
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Inactivation of the heme degrading enzyme IsdI by an active site substitution that diminishes heme ruffling.
J.Biol.Chem., 287, 2012
4K4X
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BU of 4k4x by Molmil
Coxsackievirus B3 polymerase elongation complex (r2_form), rna
分子名称: GLYCEROL, MAGNESIUM ION, RNA (5'-R(*AP*AP*GP*UP*CP*UP*CP*CP*AP*GP*GP*UP*CP*UP*CP*UP*CP*GP*UP*CP*GP*AP*AP*A)-3'), ...
著者Gong, P, Peersen, O.B.
登録日2013-04-12
公開日2013-05-22
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.37 Å)
主引用文献Structures of coxsackievirus, rhinovirus, and poliovirus polymerase elongation complexes solved by engineering RNA mediated crystal contacts.
Plos One, 8, 2013
1TO1
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BU of 1to1 by Molmil
crystal structure of the complex of subtilisin BPN' with chymotrypsin inhibitor 2 Y61A mutant
分子名称: CALCIUM ION, CITRIC ACID, PENTAETHYLENE GLYCOL, ...
著者Radisky, E.S, Kwan, G, Karen Lu, C.J, Koshland Jr, D.E.
登録日2004-06-11
公開日2004-11-09
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献Binding, Proteolytic, and Crystallographic Analyses of Mutations at the Protease-Inhibitor Interface of the Subtilisin BPN'/Chymotrypsin Inhibitor 2 Complex(,).
Biochemistry, 43, 2004
1TO2
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BU of 1to2 by Molmil
crystal structure of the complex of subtilisin BPN' with chymotrypsin inhibitor 2 M59K, in pH 9 cryosoak
分子名称: CALCIUM ION, CITRIC ACID, POLYETHYLENE GLYCOL (N=34), ...
著者Radisky, E.S, Kwan, G, Karen Lu, C.J, Koshland Jr, D.E.
登録日2004-06-11
公開日2004-11-09
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Binding, Proteolytic, and Crystallographic Analyses of Mutations at the Protease-Inhibitor Interface of the Subtilisin BPN'/Chymotrypsin Inhibitor 2 Complex(,).
Biochemistry, 43, 2004
1DD7
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BU of 1dd7 by Molmil
MURINE INDUCIBLE NITRIC OXIDE SYNTHASE OXYGENASE DOMAIN (DELTA 114) (N-[(1,3-BENZODIOXOL-5-YL)METHYL]-1-[2-(1H-IMIDAZOL-1-YL)PYRIMIDIN-4-YL]-4-(METHOXYCARBONYL)-PIPERAZINE-2-ACETAMIDE COMPLEX
分子名称: INDUCIBLE NITRIC OXIDE SYNTHASE, PROTOPORPHYRIN IX CONTAINING FE, SULFITE ION, ...
著者Adler, M, Whitlow, M.
登録日1999-11-08
公開日2000-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Allosteric inhibitors of inducible nitric oxide synthase dimerization discovered via combinatorial chemistry.
Proc.Natl.Acad.Sci.USA, 97, 2000
4KKO
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BU of 4kko by Molmil
Crystal Structure of HIV-1 Reverse Transcriptase in Complex with 4-((4-methoxy-6-(2-morpholinoethoxy)-1,3,5-triazin-2-yl)amino)-2-((3-methylbut-2-en-1-yl)oxy)benzonitrile (JLJ513), a non-nucleoside inhibitor
分子名称: 4-({4-methoxy-6-[2-(morpholin-4-yl)ethoxy]-1,3,5-triazin-2-yl}amino)-2-(3-methylbutoxy)benzonitrile, HIV-1 reverse transcriptase, p51 subunit, ...
著者Frey, K.M, Anderson, K.S.
登録日2013-05-06
公開日2013-08-14
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.89 Å)
主引用文献Extension into the entrance channel of HIV-1 reverse transcriptase-Crystallography and enhanced solubility.
Bioorg.Med.Chem.Lett., 23, 2013
4K50
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BU of 4k50 by Molmil
Rhinovirus 16 polymerase elongation complex (r1_form)
分子名称: ACETATE ION, GLYCEROL, RNA (33-MER), ...
著者Gong, P, Peersen, O.B.
登録日2013-04-12
公開日2013-05-22
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.93 Å)
主引用文献Structures of coxsackievirus, rhinovirus, and poliovirus polymerase elongation complexes solved by engineering RNA mediated crystal contacts.
Plos One, 8, 2013
2XU4
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BU of 2xu4 by Molmil
CATHEPSIN L WITH A NITRILE INHIBITOR
分子名称: (2S,4R)-4-(2-chlorophenyl)sulfonyl-1-[1-(4-fluorophenyl)cyclopropyl]carbonyl-N-[1-(iminomethyl)cyclopropyl]pyrrolidine-2-carboxamide, CATHEPSIN L1, GLYCEROL
著者Banner, D.W, Benz, J.M, Haap, W.
登録日2010-10-14
公開日2011-01-12
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.12 Å)
主引用文献Systematic Investigation of Halogen Bonding in Protein-Ligand Interactions.
Angew.Chem.Int.Ed.Engl., 50, 2011
1USQ
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BU of 1usq by Molmil
Complex of E. Coli DraE adhesin with Chloramphenicol
分子名称: 1,2-ETHANEDIOL, CHLORAMPHENICOL, DR HEMAGGLUTININ STRUCTURAL SUBUNIT, ...
著者Anderson, K.L, Billington, J, Pettigrew, D, Cota, E, Roversi, P, Simpson, P, Chen, H.A, Urvil, P, Dumerle, L, Barlow, P, Medof, E, Smith, R.A.G, Nowicki, B, Le Bouguenec, C, Lea, S.M, Matthews, S.
登録日2003-11-27
公開日2004-08-31
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献High Resolution Studies of the Afa/Dr Adhesin Drae and its Interaction with Chloramphenicol
J.Biol.Chem., 279, 2004
2XF4
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BU of 2xf4 by Molmil
Crystal structure of Salmonella enterica serovar typhimurium YcbL
分子名称: HYDROXYACYLGLUTATHIONE HYDROLASE, TETRAETHYLENE GLYCOL, ZINC ION
著者Stamp, A, Owen, P, El Omari, K, Nichols, C, Lockyer, M, Lamb, H, Charles, I, Hawkins, A.R, Stammers, D.K.
登録日2010-05-20
公開日2010-07-28
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structural and Functional Characterization of Salmonella Enterica Serovar Typhimurium Ycbl: An Unusual Type II Glyoxalase
Protein Sci., 19, 2010
1UT1
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BU of 1ut1 by Molmil
DraE adhesin from Escherichia Coli
分子名称: 1,2-ETHANEDIOL, DR HEMAGGLUTININ STRUCTURAL SUBUNIT, SULFATE ION
著者Anderson, K.L, Billington, J, Pettigrew, D, Cota, E, Roversi, P, Simpson, P, Chen, H.A, Urvil, P, Dumerle, L, Barlow, P, Medof, E, Smith, R.A.G, Nowicki, B, Le Bouguenec, C, Lea, S.M, Matthews, S.
登録日2003-12-02
公開日2004-08-31
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献High Resolution Studies of the Afa/Dr Adhesin Drae and its Interaction with Chloramphenicol
J.Biol.Chem., 279, 2004
1DO3
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BU of 1do3 by Molmil
CARBONMONOXY-MYOGLOBIN (MUTANT L29W) AFTER PHOTOLYSIS AT T>180K
分子名称: CARBON MONOXIDE, MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Ostermann, A, Waschipky, R, Parak, F.G, Nienhaus, G.U.
登録日1999-12-18
公開日2000-01-05
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Ligand binding and conformational motions in myoglobin.
Nature, 404, 2000
2YJF
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BU of 2yjf by Molmil
Oligomeric assembly of actin bound to MRTF-A
分子名称: ACTIN, ALPHA SKELETAL MUSCLE, ADENOSINE-5'-TRIPHOSPHATE, ...
著者Mouilleron, S, Langer, C.A, Guettler, S, McDonald, N.Q, Treisman, R.
登録日2011-05-19
公開日2011-07-06
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Structure of a pentavalent G-actin*MRTF-A complex reveals how G-actin controls nucleocytoplasmic shuttling of a transcriptional coactivator.
Sci Signal, 4, 2011
1SIB
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BU of 1sib by Molmil
REFINED CRYSTAL STRUCTURES OF SUBTILISIN NOVO IN COMPLEX WITH WILD-TYPE AND TWO MUTANT EGLINS. COMPARISON WITH OTHER SERINE PROTEINASE INHIBITOR COMPLEXES
分子名称: CALCIUM ION, EGLIN C, SUBTILISIN NOVO BPN'
著者Gruetter, M.G, Heinz, D.W, Priestle, J.P.
登録日1993-08-02
公開日1993-10-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Refined crystal structures of subtilisin novo in complex with wild-type and two mutant eglins. Comparison with other serine proteinase inhibitor complexes.
J.Mol.Biol., 217, 1991
1DLV
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BU of 1dlv by Molmil
BIOSYNTHETIC THIOLASE FROM ZOOGLOEA RAMIGERA IN COMPLEX WITH COA
分子名称: BIOSYNTHETIC THIOLASE, COENZYME A, SULFATE ION
著者Modis, Y, Wierenga, R.K.
登録日1999-12-12
公開日2000-04-24
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献Crystallographic analysis of the reaction pathway of Zoogloea ramigera biosynthetic thiolase.
J.Mol.Biol., 297, 2000
1DO7
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BU of 1do7 by Molmil
CARBONMONOXY-MYOGLOBIN (MUTANT L29W) REBINDING STRUCTURE AFTER PHOTOLYSIS AT T< 180K
分子名称: CARBON MONOXIDE, MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Ostermann, A, Waschipky, R, Parak, F.G, Nienhaus, G.U.
登録日1999-12-19
公開日2000-01-05
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Ligand binding and conformational motions in myoglobin.
Nature, 404, 2000

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