3TGH
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![BU of 3tgh by Molmil](/molmil-images/mine/3tgh) | GAP50 the anchor in the inner membrane complex of Plasmodium | 分子名称: | COBALT (II) ION, DIMETHYL SULFOXIDE, Glideosome-associated protein 50, ... | 著者 | Bosch, J, Paige, M.H, Vaidya, A, Bergman, L, Hol, W.G.J. | 登録日 | 2011-08-17 | 公開日 | 2012-03-07 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of GAP50, the anchor of the invasion machinery in the inner membrane complex of Plasmodium falciparum. J.Struct.Biol., 178, 2012
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5C1V
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![BU of 5c1v by Molmil](/molmil-images/mine/5c1v) | CRYSTAL STRUCTURE ANALYSIS OF CATALYTIC SUBUNIT OF HUMAN CALCINEURIN | 分子名称: | FE (III) ION, PHOSPHATE ION, Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoform, ... | 著者 | Guasch, A, Fita, I, Perez-Luque, R, Aparicio, D, Aranguren-Ibanez, A, Perez-Riba, M. | 登録日 | 2015-06-15 | 公開日 | 2016-02-03 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.35 Å) | 主引用文献 | Calcineurin Undergoes a Conformational Switch Evoked via Peptidyl-Prolyl Isomerization. Plos One, 10, 2015
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7SS6
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![BU of 7ss6 by Molmil](/molmil-images/mine/7ss6) | Structure of Klebsiella LpxH in complex with JH-LPH-45 | 分子名称: | 1,2-ETHANEDIOL, 5-{4-[3-chloro-5-(trifluoromethyl)phenyl]piperazine-1-sulfonyl}-N-[5-(hydroxyamino)-5-oxopentyl]-2,3-dihydro-1H-indole-1-carboxamide, MANGANESE (II) ION, ... | 著者 | Cho, J, Cochrane, C.S, Zhou, P. | 登録日 | 2021-11-09 | 公開日 | 2023-04-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Development of LpxH Inhibitors Chelating the Active Site Dimanganese Metal Cluster of LpxH. Chemmedchem, 18, 2023
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7SS7
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![BU of 7ss7 by Molmil](/molmil-images/mine/7ss7) | Crystal structure of Klebsiella LpxH in complex with JH-LPH-50 | 分子名称: | 1,2-ETHANEDIOL, 6-{[(4-{4-[3-chloro-5-(trifluoromethyl)phenyl]piperazine-1-sulfonyl}phenyl)carbamoyl]amino}-N-hydroxyhexanamide, MANGANESE (II) ION, ... | 著者 | Cho, J, Cochrane, C.S, Zhou, P. | 登録日 | 2021-11-09 | 公開日 | 2023-04-12 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Development of LpxH Inhibitors Chelating the Active Site Dimanganese Metal Cluster of LpxH. Chemmedchem, 18, 2023
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3RL3
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![BU of 3rl3 by Molmil](/molmil-images/mine/3rl3) | Rat metallophosphodiesterase MPPED2 | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, GUANOSINE-5'-MONOPHOSPHATE, ... | 著者 | Podobnik, M, Dermol, U. | 登録日 | 2011-04-19 | 公開日 | 2011-08-10 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Unique utilization of a phosphoprotein phosphatase fold by a mammalian phosphodiesterase associated with WAGR syndrome. J.Mol.Biol., 412, 2011
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3RL4
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![BU of 3rl4 by Molmil](/molmil-images/mine/3rl4) | Rat metallophosphodiesterase MPPED2 G252H Mutant | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, GUANOSINE-5'-MONOPHOSPHATE, ... | 著者 | Podobnik, M, Dermol, U. | 登録日 | 2011-04-19 | 公開日 | 2011-08-10 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.29 Å) | 主引用文献 | Unique utilization of a phosphoprotein phosphatase fold by a mammalian phosphodiesterase associated with WAGR syndrome. J.Mol.Biol., 412, 2011
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6WII
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![BU of 6wii by Molmil](/molmil-images/mine/6wii) | Crystal structure of the K. pneumoniae LpxH/JH-LPH-41 complex | 分子名称: | 5-({[4-({4-[3-chloro-5-(trifluoromethyl)phenyl]piperazin-1-yl}sulfonyl)phenyl]carbamoyl}amino)-N-hydroxypentanamide, DIMETHYL SULFOXIDE, GLYCEROL, ... | 著者 | Cochrane, C.S, Cho, J, Fenton, B.A, Zhou, P. | 登録日 | 2020-04-09 | 公開日 | 2020-07-29 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Synthesis and evaluation of sulfonyl piperazine LpxH inhibitors. Bioorg.Chem., 102, 2020
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2HY1
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![BU of 2hy1 by Molmil](/molmil-images/mine/2hy1) | Crystal structure of Rv0805 | 分子名称: | FE (III) ION, MANGANESE (II) ION, PHOSPHATE ION, ... | 著者 | Shenoy, A.R, Capuder, M, Draskovic, P, Lamba, D, Visweswariah, S.S, Podobnik, M. | 登録日 | 2006-08-04 | 公開日 | 2006-12-26 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.932 Å) | 主引用文献 | Structural and Biochemical Analysis of the Rv0805 Cyclic Nucleotide Phosphodiesterase from Mycobacterium tuberculosis. J.Mol.Biol., 365, 2007
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5B4A
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![BU of 5b4a by Molmil](/molmil-images/mine/5b4a) | Crystal structure of LpxH with lipid X in spacegroup P21 | 分子名称: | (R)-((2R,3S,4R,5R,6R)-3-HYDROXY-2-(HYDROXYMETHYL)-5-((R)-3-HYDROXYTETRADECANAMIDO)-6-(PHOSPHONOOXY)TETRAHYDRO-2H-PYRAN-4-YL) 3-HYDROXYTETRADECANOATE, GLYCEROL, UDP-2,3-diacylglucosamine hydrolase | 著者 | Okada, C, Wakabayashi, H, Yao, M, Tanaka, I. | 登録日 | 2016-04-03 | 公開日 | 2016-09-28 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | Crystal structures of the UDP-diacylglucosamine pyrophosphohydrase LpxH from Pseudomonas aeruginosa Sci Rep, 6, 2016
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3RL5
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![BU of 3rl5 by Molmil](/molmil-images/mine/3rl5) | Rat metallophosphodiesterase MPPED2 H67R Mutant | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, Metallophosphoesterase MPPED2, ... | 著者 | Podobnik, M, Dermol, U. | 登録日 | 2011-04-19 | 公開日 | 2011-08-10 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.26 Å) | 主引用文献 | Unique utilization of a phosphoprotein phosphatase fold by a mammalian phosphodiesterase associated with WAGR syndrome. J.Mol.Biol., 412, 2011
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2KKN
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![BU of 2kkn by Molmil](/molmil-images/mine/2kkn) | Solution NMR structure of Themotoga maritima protein TM1076: Northeast Structural Genomics Consortium target VT57 | 分子名称: | Uncharacterized protein | 著者 | Cort, J.R, Yee, A, Garcia, M, Isern, N.G, Arrowsmith, C.H, Montelione, G.T, Kennedy, M.A, Northeast Structural Genomics Consortium (NESG) | 登録日 | 2009-06-26 | 公開日 | 2009-10-06 | 最終更新日 | 2024-05-08 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution NMR structure of Themotoga maritima protein TM1076 To be Published
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5B4B
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![BU of 5b4b by Molmil](/molmil-images/mine/5b4b) | Crystal structure of LpxH with lipid X in spacegroup C2 | 分子名称: | (R)-((2R,3S,4R,5R,6R)-3-HYDROXY-2-(HYDROXYMETHYL)-5-((R)-3-HYDROXYTETRADECANAMIDO)-6-(PHOSPHONOOXY)TETRAHYDRO-2H-PYRAN-4-YL) 3-HYDROXYTETRADECANOATE, GLYCEROL, UDP-2,3-diacylglucosamine hydrolase | 著者 | Okada, C, Wakabayashi, H, Yao, M, Tanaka, I. | 登録日 | 2016-04-03 | 公開日 | 2016-09-28 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Crystal structures of the UDP-diacylglucosamine pyrophosphohydrase LpxH from Pseudomonas aeruginosa Sci Rep, 6, 2016
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2HYO
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![BU of 2hyo by Molmil](/molmil-images/mine/2hyo) | Crystal structure of Rv0805 N97A mutant | 分子名称: | FE (III) ION, MANGANESE (II) ION, Rv0805N97A | 著者 | Shenoy, A.R, Capuder, M, Draskovic, P, Lamba, D, Visweswariah, S.S, Podobnik, M. | 登録日 | 2006-08-07 | 公開日 | 2006-12-26 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Structural and Biochemical Analysis of the Rv0805 Cyclic Nucleotide Phosphodiesterase from Mycobacterium tuberculosis. J.Mol.Biol., 365, 2007
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2HYP
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![BU of 2hyp by Molmil](/molmil-images/mine/2hyp) | Crystal structure of Rv0805 D66A mutant | 分子名称: | BROMIDE ION, CACODYLATE ION, FE (III) ION, ... | 著者 | Shenoy, A.R, Capuder, M, Draskovic, P, Lamba, D, Visweswariah, S.S, Podobnik, M. | 登録日 | 2006-08-07 | 公開日 | 2006-12-26 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Structural and Biochemical Analysis of the Rv0805 Cyclic Nucleotide Phosphodiesterase from Mycobacterium tuberculosis. J.Mol.Biol., 365, 2007
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2JOG
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![BU of 2jog by Molmil](/molmil-images/mine/2jog) | Structure of the calcineurin-NFAT complex | 分子名称: | Calmodulin-dependent calcineurin A subunit alpha isoform, NFAT | 著者 | Takeuchi, K, Roehrl, M.H, Sun, Z.Y, Wagner, G. | 登録日 | 2007-03-10 | 公開日 | 2007-05-22 | 最終更新日 | 2023-12-20 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure of the Calcineurin-NFAT Complex: Defining a T Cell Activation Switch Using Solution NMR and Crystal Coordinates. Structure, 15, 2007
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2ZO9
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![BU of 2zo9 by Molmil](/molmil-images/mine/2zo9) | Malonate-bound structure of the glycerophosphodiesterase from Enterobacter aerogenes (GpdQ) and characterization of the native Fe2+ metal ion preference | 分子名称: | FE (II) ION, MALONATE ION, Phosphohydrolase | 著者 | Jackson, C.J, Carr, P.D, Ollis, D.L. | 登録日 | 2008-05-07 | 公開日 | 2008-10-07 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Malonate-bound structure of the glycerophosphodiesterase from Enterobacter aerogenes (GpdQ) and characterization of the native Fe2+ metal-ion preference. Acta Crystallogr.,Sect.F, 64, 2008
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2ZOA
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![BU of 2zoa by Molmil](/molmil-images/mine/2zoa) | Malonate-bound structure of the glycerophosphodiesterase from Enterobacter aerogenes (GpdQ) COLLECTED AT 1.280 ANGSTROM | 分子名称: | FE (II) ION, MALONATE ION, Phosphohydrolase | 著者 | Ollis, D.L, Jackson, C.J, Carr, P.D. | 登録日 | 2008-05-07 | 公開日 | 2008-10-07 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Malonate-bound structure of the glycerophosphodiesterase from Enterobacter aerogenes (GpdQ) and characterization of the native Fe2+ metal-ion preference. Acta Crystallogr.,Sect.F, 64, 2008
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3AUZ
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![BU of 3auz by Molmil](/molmil-images/mine/3auz) | Crystal structure of Mre11 with manganese | 分子名称: | DNA double-strand break repair protein mre11, GLYCEROL, MANGANESE (II) ION | 著者 | Park, Y.B, Cho, Y. | 登録日 | 2011-02-18 | 公開日 | 2011-05-25 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (3.206 Å) | 主引用文献 | Crystal Structure of the Mre11-Rad50-ATP S Complex: Understanding the Interplay between Mre11 and Rad50 To be Published
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2ZBM
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![BU of 2zbm by Molmil](/molmil-images/mine/2zbm) | Crystal Structure of I115M Mutant Cold-Active Protein Tyrosine Phosphatase | 分子名称: | Protein-tyrosine-phosphatase, ZINC ION | 著者 | Tsuruta, H, Mikami, B, Yamamoto, C, Yamagata, H. | 登録日 | 2007-10-24 | 公開日 | 2008-07-29 | 最終更新日 | 2021-11-10 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | The role of group bulkiness in the catalytic activity of psychrophile cold-active protein tyrosine phosphatase Febs J., 275, 2008
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2Z72
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![BU of 2z72 by Molmil](/molmil-images/mine/2z72) | New Structure Of Cold-Active Protein Tyrosine Phosphatase At 1.1 Angstrom | 分子名称: | Protein-tyrosine-phosphatase, ZINC ION | 著者 | Tsuruta, H, Mikami, B, Yamamoto, C, Yamagata, H. | 登録日 | 2007-08-10 | 公開日 | 2008-07-29 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.1 Å) | 主引用文献 | The role of group bulkiness in the catalytic activity of psychrophile cold-active protein tyrosine phosphatase Febs J., 275, 2008
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3D03
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![BU of 3d03 by Molmil](/molmil-images/mine/3d03) | 1.9A structure of Glycerophoshphodiesterase (GpdQ) from Enterobacter aerogenes | 分子名称: | COBALT (II) ION, Phosphohydrolase | 著者 | Hadler, K.S, Tanifum, E, Yip, S.H.-C, Miti, N, Guddat, L.W, Jackson, C.J, Gahan, L.R, Carr, P.D, Nguyen, K, Ollis, D.L, Hengge, A.C, Larrabee, J.A, Schenk, G. | 登録日 | 2008-04-30 | 公開日 | 2008-10-14 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Substrate-promoted formation of a catalytically competent binuclear center and regulation of reactivity in a glycerophosphodiesterase from Enterobacter aerogenes. J.Am.Chem.Soc., 130, 2008
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3IB7
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![BU of 3ib7 by Molmil](/molmil-images/mine/3ib7) | Crystal structure of full length Rv0805 | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ACETATE ION, ... | 著者 | Podobnik, M, Dermol, U. | 登録日 | 2009-07-15 | 公開日 | 2009-09-29 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | A mycobacterial cyclic AMP phosphodiesterase that moonlights as a modifier of cell wall permeability J.Biol.Chem., 284, 2009
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3IB8
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![BU of 3ib8 by Molmil](/molmil-images/mine/3ib8) | Crystal structure of full length Rv0805 in complex with 5'-AMP | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ACETATE ION, ... | 著者 | Podobnik, M, Dermol, U. | 登録日 | 2009-07-15 | 公開日 | 2009-09-29 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | A mycobacterial cyclic AMP phosphodiesterase that moonlights as a modifier of cell wall permeability J.Biol.Chem., 284, 2009
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3JYF
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![BU of 3jyf by Molmil](/molmil-images/mine/3jyf) | The crystal structure of a 2,3-cyclic nucleotide 2-phosphodiesterase/3-nucleotidase bifunctional periplasmic precursor protein from Klebsiella pneumoniae subsp. pneumoniae MGH 78578 | 分子名称: | 2',3'-cyclic nucleotide 2'-phosphodiesterase/3'-nucleotidase bifunctional periplasmic protein, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, GLYCEROL, ... | 著者 | Fan, Y, Volkart, L, Cobb, G, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2009-09-21 | 公開日 | 2009-09-29 | 最終更新日 | 2017-11-01 | 実験手法 | X-RAY DIFFRACTION (2.43 Å) | 主引用文献 | The crystal structure of a 2,3-cyclic nucleotide 2-phosphodiesterase/3-nucleotidase bifunctional periplasmic precursor protein from Klebsiella pneumoniae subsp. pneumoniae MGH 78578 To be Published
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6NVP
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![BU of 6nvp by Molmil](/molmil-images/mine/6nvp) | |