5SS0
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![BU of 5ss0 by Molmil](/molmil-images/mine/5ss0) | |
5SRZ
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![BU of 5srz by Molmil](/molmil-images/mine/5srz) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5281440906 - (R,S) and (S,R) isomers | 分子名称: | (1R,2S)-2-[(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)amino]cyclohexane-1-carboxylic acid, (1S,2R)-2-[(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)amino]cyclohexane-1-carboxylic acid, Non-structural protein 3 | 著者 | Correy, G.J, Fraser, J.S. | 登録日 | 2022-06-09 | 公開日 | 2022-07-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SS8
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![BU of 5ss8 by Molmil](/molmil-images/mine/5ss8) | |
5SSB
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![BU of 5ssb by Molmil](/molmil-images/mine/5ssb) | |
5SSG
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![BU of 5ssg by Molmil](/molmil-images/mine/5ssg) | |
5SQ4
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![BU of 5sq4 by Molmil](/molmil-images/mine/5sq4) | |
5SSK
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![BU of 5ssk by Molmil](/molmil-images/mine/5ssk) | |
5SRH
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![BU of 5srh by Molmil](/molmil-images/mine/5srh) | |
5SQI
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![BU of 5sqi by Molmil](/molmil-images/mine/5sqi) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5016127255 - (R,R) and (S,S) isomers | 分子名称: | (1R,2R)-4-hydroxy-1-[4-(methylcarbamamido)benzamido]-2,3-dihydro-1H-indene-2-carboxylic acid, (1S,2S)-4-hydroxy-1-[4-(methylcarbamamido)benzamido]-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 | 著者 | Correy, G.J, Fraser, J.S. | 登録日 | 2022-06-09 | 公開日 | 2022-07-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRP
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5SR1
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![BU of 5sr1 by Molmil](/molmil-images/mine/5sr1) | |
5SS1
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![BU of 5ss1 by Molmil](/molmil-images/mine/5ss1) | |
5SR5
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![BU of 5sr5 by Molmil](/molmil-images/mine/5sr5) | |
5SSA
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![BU of 5ssa by Molmil](/molmil-images/mine/5ssa) | |
5SPZ
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![BU of 5spz by Molmil](/molmil-images/mine/5spz) | |
5SSH
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![BU of 5ssh by Molmil](/molmil-images/mine/5ssh) | |
5SRK
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![BU of 5srk by Molmil](/molmil-images/mine/5srk) | |
5SQ2
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![BU of 5sq2 by Molmil](/molmil-images/mine/5sq2) | |
5SRW
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![BU of 5srw by Molmil](/molmil-images/mine/5srw) | |
5SQ9
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![BU of 5sq9 by Molmil](/molmil-images/mine/5sq9) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5010894420 - (R,R) and (S,S) isomers | 分子名称: | (1R,2R)-4-hydroxy-1-{4-[(propan-2-yl)carbamamido]benzamido}-2,3-dihydro-1H-indene-2-carboxylic acid, (1S,2S)-4-hydroxy-1-{4-[(propan-2-yl)carbamamido]benzamido}-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 | 著者 | Correy, G.J, Fraser, J.S. | 登録日 | 2022-06-09 | 公開日 | 2022-07-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SS3
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![BU of 5ss3 by Molmil](/molmil-images/mine/5ss3) | |
5SQB
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![BU of 5sqb by Molmil](/molmil-images/mine/5sqb) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5010894390 - (R,R) and (S,S) isomers | 分子名称: | (1R,2R)-1-({6-[(cyclopropylmethyl)amino]pyridine-3-carbonyl}amino)-4-hydroxy-2,3-dihydro-1H-indene-2-carboxylic acid, (1S,2S)-1-({6-[(cyclopropylmethyl)amino]pyridine-3-carbonyl}amino)-4-hydroxy-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 | 著者 | Correy, G.J, Fraser, J.S. | 登録日 | 2022-06-09 | 公開日 | 2022-07-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SSI
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![BU of 5ssi by Molmil](/molmil-images/mine/5ssi) | |
5SSN
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![BU of 5ssn by Molmil](/molmil-images/mine/5ssn) | |
5SQL
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![BU of 5sql by Molmil](/molmil-images/mine/5sql) | |