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PDB: 33 件

6G48
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Sporosarcina pasteurii urease inhibited by silver
分子名称: 1,2-ETHANEDIOL, HYDROXIDE ION, NICKEL (II) ION, ...
著者Mazzei, L, Cianci, M, Ciurli, S.
登録日2018-03-27
公開日2019-01-16
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献The structure of urease inactivated by Ag(i): a new paradigm for enzyme inhibition by heavy metals.
Dalton Trans, 47, 2018
7B5A
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X-ray crystal structure of Sporosarcina pasteurii urease inhibited by Ag(PEt3)2NO3 determined at 1.97 Angstroms
分子名称: 1,2-ETHANEDIOL, NICKEL (II) ION, OXYGEN ATOM, ...
著者Mazzei, L, Cianci, M, Ciurli, S.
登録日2020-12-03
公開日2021-10-13
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Kinetic and structural analysis of the inactivation of urease by mixed-ligand phosphine halide Ag(I) complexes.
J.Inorg.Biochem., 218, 2021
2UBP
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STRUCTURE OF NATIVE UREASE FROM BACILLUS PASTEURII
分子名称: NICKEL (II) ION, PROTEIN (UREASE ALPHA SUBUNIT), PROTEIN (UREASE BETA SUBUNIT), ...
著者Benini, S, Rypniewski, W.R, Wilson, K.S, Ciurli, S, Mangani, S.
登録日1998-11-04
公開日1999-11-08
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A new proposal for urease mechanism based on the crystal structures of the native and inhibited enzyme from Bacillus pasteurii: why urea hydrolysis costs two nickels.
Structure Fold.Des., 7, 1999
3UBP
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DIAMIDOPHOSPHATE INHIBITED BACILLUS PASTEURII UREASE
分子名称: DIAMIDOPHOSPHATE, NICKEL (II) ION, PROTEIN (UREASE ALPHA SUBUNIT), ...
著者Benini, S, Rypniewski, W.R, Wilson, K.S, Miletti, S, Mangani, S, Ciurli, S.
登録日1998-12-16
公開日1999-12-17
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A new proposal for urease mechanism based on the crystal structures of the native and inhibited enzyme from Bacillus pasteurii: why urea hydrolysis costs two nickels.
Structure Fold.Des., 7, 1999
5FSE
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2.07 A resolution 1,4-Benzoquinone inhibited Sporosarcina pasteurii urease
分子名称: 1,2-ETHANEDIOL, HYDROXIDE ION, NICKEL (II) ION, ...
著者Mazzei, L, Cianci, M, Musiani, F, Ciurli, S.
登録日2016-01-04
公開日2016-03-23
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献Inactivation of Urease by 1,4-Benzoquinone: Chemistry at the Protein Surface.
Dalton Trans, 45, 2016
1S3T
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BORATE INHIBITED BACILLUS PASTEURII UREASE CRYSTAL STRUCTURE
分子名称: BORIC ACID, NICKEL (II) ION, SULFATE ION, ...
著者Benini, S, Rypniewski, W.R, Wilson, K.S, Ciurli, S, Mangani, S.
登録日2004-01-14
公開日2004-04-06
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Molecular Details of Urease Inhibition by Boric Acid: Insights into the Catalytic Mechanism.
J.Am.Chem.Soc., 126, 2004
6I9Y
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The 2.14 A X-ray crystal structure of Sporosarcina pasteurii urease in complex with Au(I) ions
分子名称: 1,2-ETHANEDIOL, GOLD ION, HYDROXIDE ION, ...
著者Mazzei, L, Cianci, M, Ciurli, S.
登録日2018-11-26
公開日2019-05-01
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Inhibition Mechanism of Urease by Au(III) Compounds Unveiled by X-ray Diffraction Analysis.
Acs Med.Chem.Lett., 10, 2019
6ZO0
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2.23 A resolution 3,4-dimethylcatechol (3,4-dimethylbenzene-1,2-diol) inhibited Sporosarcina pasteurii urease
分子名称: 1,2-ETHANEDIOL, HYDROXIDE ION, NICKEL (II) ION, ...
著者Mazzei, L, Cianci, M, Musiani, F, Ciurli, S.
登録日2020-07-07
公開日2020-12-23
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献Inhibition of Urease, a Ni-Enzyme: The Reactivity of a Key Thiol With Mono- and Di-Substituted Catechols Elucidated by Kinetic, Structural, and Theoretical Studies.
Angew.Chem.Int.Ed.Engl., 60, 2021
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