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PDB: 1 件

4YU2
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Crystal structure of DYRK1A with harmine-derivatized AnnH-75 inhibitor
分子名称: (1-chloro-7-methoxy-9H-beta-carbolin-9-yl)acetonitrile, Dual specificity tyrosine-phosphorylation-regulated kinase 1A, SULFATE ION, ...
著者Chaikuad, A, Wurzlbauer, A, Nowak, R, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Bracher, F, Knapp, S, Structural Genomics Consortium (SGC)
登録日2015-03-18
公開日2015-03-25
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献How to Separate Kinase Inhibition from Undesired Monoamine Oxidase A Inhibition-The Development of the DYRK1A Inhibitor AnnH75 from the Alkaloid Harmine.
Molecules, 25, 2020

238582

件を2025-07-09に公開中

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