9MVP
 
 | Crystal Structure of SARS-CoV-2 Main Protease (Mpro)in Complex with Inhibitor AVI-4516 | 分子名称: | (3M,5P)-5-(1H-1,2,3-benzotriazol-1-yl)-3-(isoquinolin-4-yl)-6-methyl-1-(prop-2-en-1-yl)pyrimidine-2,4(1H,3H)-dione, 1,2-ETHANEDIOL, 3C-like proteinase nsp5 | 著者 | Diallo, A, Gumpena, R, Verba, K. | 登録日 | 2025-01-15 | 公開日 | 2025-07-23 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus M Pro inhibitors with potent in vivo efficacy. Sci Adv, 11, 2025
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9MVQ
 
 | Crystal Structure of SARS-CoV-2 Main Protease (Mpro) variant Q192T in Complex with Inhibitor AVI-4303 | 分子名称: | (3M,5P,6M)-5-(1H-1,2,3-benzotriazol-1-yl)-6-(3-chlorophenyl)-3-(isoquinolin-4-yl)pyrimidine-2,4(1H,3H)-dione, 1,2-ETHANEDIOL, 3C-like proteinase nsp5, ... | 著者 | Diallo, A, Gumpena, R, Partridge, J, Verba, K. | 登録日 | 2025-01-15 | 公開日 | 2025-07-23 | 実験手法 | X-RAY DIFFRACTION (1.57 Å) | 主引用文献 | Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus M Pro inhibitors with potent in vivo efficacy. Sci Adv, 11, 2025
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9MVO
 
 | Crystal Structure of SARS-CoV-2 Main Protease (Mpro) in Complex with Inhibitor AVI-4692 | 分子名称: | (3M,5P,6M)-5-(1H-1,2,3-benzotriazol-1-yl)-6-(3-chlorophenyl)-3-(isoquinolin-4-yl)-1-(prop-2-en-1-yl)pyrimidine-2,4(1H,3H)-dione, (3M,5P,6M)-5-(1H-1,2,3-benzotriazol-1-yl)-6-(3-chlorophenyl)-3-(isoquinolin-4-yl)-1-(prop-2-yn-1-yl)pyrimidine-2,4(1H,3H)-dione, 3C-like proteinase nsp5 | 著者 | Diallo, A, Gumpena, R, Verba, K. | 登録日 | 2025-01-15 | 公開日 | 2025-07-23 | 最終更新日 | 2025-08-13 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus M Pro inhibitors with potent in vivo efficacy. Sci Adv, 11, 2025
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9MVM
 
 | Crystal Structure of SARS-CoV-2 Main Protease (Mpro)in Complex with Inhibitor AVI-3318 | 分子名称: | 1-[(4-chlorothiophen-2-yl)methyl]-3-[(2-oxo-1,2-dihydropyridin-3-yl)methyl]-1,3-diazinane-2,4-dione, Replicase polyprotein 1ab | 著者 | Diallo, A, Gumpena, R, Verba, K. | 登録日 | 2025-01-15 | 公開日 | 2025-07-23 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus M Pro inhibitors with potent in vivo efficacy. Sci Adv, 11, 2025
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