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PDB: 4 件

9MVP
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BU of 9mvp by Molmil
Crystal Structure of SARS-CoV-2 Main Protease (Mpro)in Complex with Inhibitor AVI-4516
分子名称: (3M,5P)-5-(1H-1,2,3-benzotriazol-1-yl)-3-(isoquinolin-4-yl)-6-methyl-1-(prop-2-en-1-yl)pyrimidine-2,4(1H,3H)-dione, 1,2-ETHANEDIOL, 3C-like proteinase nsp5
著者Diallo, A, Gumpena, R, Verba, K.
登録日2025-01-15
公開日2025-07-23
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus M Pro inhibitors with potent in vivo efficacy.
Sci Adv, 11, 2025
9MVQ
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BU of 9mvq by Molmil
Crystal Structure of SARS-CoV-2 Main Protease (Mpro) variant Q192T in Complex with Inhibitor AVI-4303
分子名称: (3M,5P,6M)-5-(1H-1,2,3-benzotriazol-1-yl)-6-(3-chlorophenyl)-3-(isoquinolin-4-yl)pyrimidine-2,4(1H,3H)-dione, 1,2-ETHANEDIOL, 3C-like proteinase nsp5, ...
著者Diallo, A, Gumpena, R, Partridge, J, Verba, K.
登録日2025-01-15
公開日2025-07-23
実験手法X-RAY DIFFRACTION (1.57 Å)
主引用文献Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus M Pro inhibitors with potent in vivo efficacy.
Sci Adv, 11, 2025
9MVO
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BU of 9mvo by Molmil
Crystal Structure of SARS-CoV-2 Main Protease (Mpro) in Complex with Inhibitor AVI-4692
分子名称: (3M,5P,6M)-5-(1H-1,2,3-benzotriazol-1-yl)-6-(3-chlorophenyl)-3-(isoquinolin-4-yl)-1-(prop-2-en-1-yl)pyrimidine-2,4(1H,3H)-dione, (3M,5P,6M)-5-(1H-1,2,3-benzotriazol-1-yl)-6-(3-chlorophenyl)-3-(isoquinolin-4-yl)-1-(prop-2-yn-1-yl)pyrimidine-2,4(1H,3H)-dione, 3C-like proteinase nsp5
著者Diallo, A, Gumpena, R, Verba, K.
登録日2025-01-15
公開日2025-07-23
最終更新日2025-08-13
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus M Pro inhibitors with potent in vivo efficacy.
Sci Adv, 11, 2025
9MVM
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BU of 9mvm by Molmil
Crystal Structure of SARS-CoV-2 Main Protease (Mpro)in Complex with Inhibitor AVI-3318
分子名称: 1-[(4-chlorothiophen-2-yl)methyl]-3-[(2-oxo-1,2-dihydropyridin-3-yl)methyl]-1,3-diazinane-2,4-dione, Replicase polyprotein 1ab
著者Diallo, A, Gumpena, R, Verba, K.
登録日2025-01-15
公開日2025-07-23
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus M Pro inhibitors with potent in vivo efficacy.
Sci Adv, 11, 2025

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件を2025-10-22に公開中

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