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PDB: 2 件

5OBJ
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BU of 5obj by Molmil
Aurora A kinase in complex with 2-(3-fluorophenyl)quinoline-4-carboxylic acid and ATP
分子名称: 2-(3-fluorophenyl)quinoline-4-carboxylic acid, ADENOSINE-5'-TRIPHOSPHATE, Aurora kinase A, ...
著者Rossmann, M, Janecek, M, Hyvonen, M.
登録日2017-06-28
公開日2017-08-09
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.901 Å)
主引用文献Computationally-guided optimization of small-molecule inhibitors of the Aurora A kinase-TPX2 protein-protein interaction.
Chem. Commun. (Camb.), 53, 2017
5OBR
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BU of 5obr by Molmil
Aurora A kinase in complex with 2-(3-chloro-5-fluorophenyl)quinoline-4-carboxylic acid and JNJ-7706621
分子名称: 2-(3-chloranyl-5-fluoranyl-phenyl)quinoline-4-carboxylic acid, 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1H-1,2,4-triazol-3-yl}amino)benzenesulfonamide, Aurora kinase A, ...
著者Rossmann, M, Janecek, M, Hyvonen, M.
登録日2017-06-29
公開日2017-08-09
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.62 Å)
主引用文献Computationally-guided optimization of small-molecule inhibitors of the Aurora A kinase-TPX2 protein-protein interaction.
Chem. Commun. (Camb.), 53, 2017

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件を2024-07-31に公開中

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