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PDB: 3 件

7XMF
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BU of 7xmf by Molmil
Cryo-EM structure of human NaV1.7/beta1/beta2-Nav1.7-IN2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 3-[[4-[3-(4-fluoranyl-2-methyl-phenoxy)azetidin-1-yl]pyrimidin-2-yl]amino]-~{N}-methyl-benzamide, ...
著者Zhang, J.T, Jiang, D.H.
登録日2022-04-25
公開日2022-11-30
最終更新日2022-12-28
実験手法ELECTRON MICROSCOPY (3.07 Å)
主引用文献Structural basis for Na V 1.7 inhibition by pore blockers.
Nat.Struct.Mol.Biol., 29, 2022
7XM9
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BU of 7xm9 by Molmil
Cryo-EM structure of human NaV1.7/beta1/beta2-XEN907
分子名称: (7~{R})-1'-pentylspiro[6~{H}-furo[3,2-f][1,3]benzodioxole-7,3'-indole]-2'-one, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者zhang, J.T, Jiang, D.H.
登録日2022-04-25
公開日2022-11-30
最終更新日2022-12-28
実験手法ELECTRON MICROSCOPY (3.22 Å)
主引用文献Structural basis for Na V 1.7 inhibition by pore blockers.
Nat.Struct.Mol.Biol., 29, 2022
7XMG
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BU of 7xmg by Molmil
Cryo-EM structure of human NaV1.7/beta1/beta2-TCN-1752
分子名称: (1~{Z})-~{N}-[2-methyl-3-[(~{E})-[6-[4-[[4-(trifluoromethyloxy)phenyl]methoxy]piperidin-1-yl]-1~{H}-1,3,5-triazin-2-ylidene]amino]phenyl]ethanimidic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Jiang, D.H, Zhang, J.T.
登録日2022-04-25
公開日2022-11-30
最終更新日2022-12-28
実験手法ELECTRON MICROSCOPY (3.09 Å)
主引用文献Structural basis for Na V 1.7 inhibition by pore blockers.
Nat.Struct.Mol.Biol., 29, 2022

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件を2024-09-04に公開中

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