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PDB: 1 件

7FIC
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Reversible lysine-targeted probes reveal residence time-based kinase selectivity in vivo
分子名称: 6-[(5-cyclopropyl-1~{H}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{N}-prop-2-ynyl-pyrimidine-4-carboxamide, Aurora kinase A, CHLORIDE ION
著者Craven, G.B, Wan, X.B, Taunton, J.
登録日2021-07-31
公開日2022-06-08
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.32 Å)
主引用文献Reversible lysine-targeted probes reveal residence time-based kinase selectivity.
Nat.Chem.Biol., 18, 2022

221051

件を2024-06-12に公開中

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