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PDB: 7 件

8X0H
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BU of 8x0h by Molmil
Human FL Metabotropic glutamate receptor 5, mGlu5-5M with quisqualate, Rcc conformation
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 5
著者Vinothkumar, K.R, Lebon, G, Cannone, G.
登録日2023-11-04
公開日2024-11-06
最終更新日2025-01-29
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Conformational diversity in class C GPCR positive allosteric modulation.
Nat Commun, 16, 2025
8X0E
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BU of 8x0e by Molmil
Human FL Metabotropic glutamate receptor 5, mGlu5-5M with agonist and PAM, W785A mutant
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 5
著者Vinothkumar, K.R, Lebon, G, Cannone, G.
登録日2023-11-04
公開日2024-11-06
最終更新日2025-01-29
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Conformational diversity in class C GPCR positive allosteric modulation.
Nat Commun, 16, 2025
8X0F
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BU of 8x0f by Molmil
Human FL Metabotropic glutamate receptor 5, mGlu5-5M with quisqualate and PAM VU29
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 5, ...
著者Vinothkumar, K.R, Lebon, G, Cannone, G.
登録日2023-11-04
公開日2024-11-06
最終更新日2025-01-29
実験手法ELECTRON MICROSCOPY (3.3 Å)
主引用文献Conformational diversity in class C GPCR positive allosteric modulation.
Nat Commun, 16, 2025
8X0B
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BU of 8x0b by Molmil
Human FL Metabotropic glutamate receptor 5, mGlu5-5M with Quisqualate and VU0424465
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 5, ...
著者Vinothkumar, K.R, Lebon, G, Cannone, G.
登録日2023-11-04
公開日2024-11-06
最終更新日2025-01-29
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Conformational diversity in class C GPCR positive allosteric modulation.
Nat Commun, 16, 2025
8X0C
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BU of 8x0c by Molmil
Human FL Metabotropic glutamate receptor 5, mGlu5-5M with quisqualate and VU0424465, conformer 1
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 5, ...
著者Vinothkumar, K.R, Lebon, G, Cannone, G.
登録日2023-11-04
公開日2024-11-06
最終更新日2025-01-29
実験手法ELECTRON MICROSCOPY (3.2 Å)
主引用文献Conformational diversity in class C GPCR positive allosteric modulation.
Nat Commun, 16, 2025
8X0G
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BU of 8x0g by Molmil
Human FL Metabotropic glutamate receptor 5, mGlu5-5M with quisqualate, Acc conformation (purified with PAM VU0409551 but not modelled)
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 5
著者Vinothkumar, K.R, Lebon, G, Cannone, G.
登録日2023-11-04
公開日2024-11-06
最終更新日2025-01-29
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Conformational diversity in class C GPCR positive allosteric modulation.
Nat Commun, 16, 2025
8X0D
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BU of 8x0d by Molmil
Human FL Metabotropic glutamate receptor 5, mGlu5-5M with quisqualate and VU0424465, conformer 2
分子名称: (S)-2-AMINO-3-(3,5-DIOXO-[1,2,4]OXADIAZOLIDIN-2-YL)-PROPIONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose, Metabotropic glutamate receptor 5, ...
著者Lebon, G, Cannone, G, Vinothkumar, K.R.
登録日2023-11-04
公開日2024-11-06
最終更新日2025-01-29
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Conformational diversity in class C GPCR positive allosteric modulation.
Nat Commun, 16, 2025

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件を2025-07-09に公開中

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