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PDB: 1 件

4YHF
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Bruton's tyrosine kinase in complex with a t-butyl cyanoacrylamide inhibitor
分子名称: (2S)-2-({(3R)-3-[4-amino-3-(4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrile, 1,2-ETHANEDIOL, CHLORIDE ION, ...
著者Paavilainen, V.O, McFarland, J.M, Taunton, J.
登録日2015-02-27
公開日2015-05-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Prolonged and tunable residence time using reversible covalent kinase inhibitors.
Nat.Chem.Biol., 11, 2015

222036

件を2024-07-03に公開中

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