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PDB: 1 件

3OG7
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B-Raf Kinase V600E oncogenic mutant in complex with PLX4032
分子名称: AKAP9-BRAF fusion protein, N-(3-{[5-(4-chlorophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide
著者Zhang, Y, Zhang, K.Y, Zhang, C.
登録日2010-08-16
公開日2010-09-22
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Clinical efficacy of a RAF inhibitor needs broad target blockade in BRAF-mutant melanoma.
Nature, 467, 2010

222926

件を2024-07-24に公開中

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