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PDB: 1 件

3ZYU
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Crystal Structure of the first bromodomain of human BRD4 in complex with I-BET151(GSK1210151A)
分子名称: 1,2-ETHANEDIOL, 7-(3,5-DIMETHYL-1,2-OXAZOL-4-YL)-8-METHOXY-1-[(1R)-1-(PYRIDIN-2-YL)ETHYL]-1H,2H,3H-IMIDAZO[4,5-C]QUINOLIN-2-ONE, BROMODOMAIN-CONTAINING PROTEIN 4
著者Chung, C.W, Mirguet, O.
登録日2011-08-25
公開日2011-11-02
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Inhibition of Bet Recruitment to Chromatin as an Effective Treatment for Mll-Fusion Leukaemia.
Nature, 478, 2011

223532

件を2024-08-07に公開中

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