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PDB: 1 件

3KB7
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Crystal structure of Polo-like kinase 1 in complex with a pyrazoloquinazoline inhibitor
分子名称: 8-{[2-methoxy-5-(4-methylpiperazin-1-yl)phenyl]amino}-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide, L(+)-TARTARIC ACID, Serine/threonine-protein kinase PLK1, ...
著者Bossi, R.T, Bertrand, J.A.
登録日2009-10-20
公開日2010-05-19
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Identification of 4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline derivatives as a new class of orally and selective Polo-like kinase 1 inhibitors
J.Med.Chem., 53, 2010

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件を2024-10-16に公開中

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