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PDB: 3 件

3BGZ
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BU of 3bgz by Molmil
Human Pim-1 kinase in complex with diphenyl indole inhibitor VX3
分子名称: 2,3-diphenyl-1H-indole-7-carboxylic acid, Proto-oncogene serine/threonine-protein kinase Pim-1
著者Jacobs, M.D.
登録日2007-11-27
公開日2007-12-11
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Docking study yields four novel inhibitors of the protooncogene pim-1 kinase.
J.Med.Chem., 51, 2008
3BGQ
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BU of 3bgq by Molmil
Human Pim-1 kinase in complex with an triazolo pyridazine inhibitor VX2
分子名称: N-cyclohexyl-3-[3-(trifluoromethyl)phenyl][1,2,4]triazolo[4,3-b]pyridazin-6-amine, Proto-oncogene serine/threonine-protein kinase Pim-1
著者Jacobs, M.D.
登録日2007-11-27
公開日2007-12-11
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Docking study yields four novel inhibitors of the protooncogene pim-1 kinase.
J.Med.Chem., 51, 2008
3BGP
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BU of 3bgp by Molmil
Human Pim-1 complexed with a benzoisoxazole inhibitor VX1
分子名称: 4-[3-(4-chlorophenyl)-2,1-benzisoxazol-5-yl]pyrimidin-2-amine, Proto-oncogene serine/threonine-protein kinase Pim-1
著者Jacobs, M.D.
登録日2007-11-27
公開日2007-12-11
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Docking study yields four novel inhibitors of the protooncogene pim-1 kinase.
J.Med.Chem., 51, 2008

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件を2024-07-31に公開中

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