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PDB: 1 件

3P9J
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Aurora A kinase domain with phthalazinone pyrazole inhibitor
分子名称: 4-[(5-methyl-1H-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2H)-one, Serine/threonine-protein kinase 6
著者Kairies, N.A, Oliveira, T, Engh, R.A.
登録日2010-10-17
公開日2011-03-23
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Phthalazinone pyrazoles as potent, selective, and orally bioavailable inhibitors of aurora-a kinase.
J.Med.Chem., 54, 2011

222415

件を2024-07-10に公開中

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