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PDB: 1 件

4Y73
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Crystal structure of IRAK4 kinase domain with inhibitor
分子名称: 5-{[(1R,2S)-2-aminocyclohexyl]amino}-N-[1-methyl-3-(trifluoromethyl)-1H-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide, Interleukin-1 receptor-associated kinase 4
著者Lesburg, C.A.
登録日2015-02-13
公開日2015-05-20
最終更新日2015-07-15
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献Discovery of 5-Amino-N-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide Inhibitors of IRAK4.
Acs Med.Chem.Lett., 6, 2015

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件を2024-08-14に公開中

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