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PDB: 1 件

7Z61
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BU of 7z61 by Molmil
Crystal structure of PI3Kgamma with a dihydropurinone inhibitor (compound 18)
分子名称: 9-[(3~{R},4~{R})-4-fluoranylpyrrolidin-3-yl]-7-methyl-2-[(7-methylquinolin-6-yl)amino]purin-8-one, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
著者Goldberg, F.W, Ting, A.K.T, Schimpl, M.
登録日2022-03-10
公開日2022-07-13
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.738 Å)
主引用文献Optimization of hERG and Pharmacokinetic Properties for Basic Dihydro-8 H -purin-8-one Inhibitors of DNA-PK.
Acs Med.Chem.Lett., 13, 2022

221051

件を2024-06-12に公開中

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