Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
PDB: 1 件

4R3C
DownloadVisualize
BU of 4r3c by Molmil
Crystal structure of p38 alpha MAP kinase in complex with a novel isoform selective drug candidate
分子名称: 4-[3-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL]PYRIDINE, 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine, CHLORIDE ION, ...
著者Grum-Tokars, V.L, Minasov, G, Roy, S.M, Anderson, W.F, Watterson, D.M.
登録日2014-08-14
公開日2015-02-25
最終更新日2017-11-22
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Targeting human central nervous system protein kinases: An isoform selective p38 alpha MAPK inhibitor that attenuates disease progression in Alzheimer's disease mouse models.
ACS Chem Neurosci, 6, 2015

222926

件を2024-07-24に公開中

PDB statisticsPDBj update infoContact PDBjnumon