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PDB: 1 件

6KG2
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BU of 6kg2 by Molmil
Human MTHFD2 in complex with Compound 18
分子名称: Bifunctional methylenetetrahydrofolate dehydrogenase/cyclohydrolase, mitochondrial, N-[2-chloranyl-4-[[7-methyl-8-(4-methylpiperazin-1-yl)-5-oxidanylidene-2,4-dihydro-1H-chromeno[3,4-c]pyridin-3-yl]carbonyl]phenyl]methanesulfonamide, ...
著者Suzuki, M, Matsui, Y, Ota, M, Kawai, J.
登録日2019-07-10
公開日2019-11-13
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Discovery of a Potent, Selective, and Orally Available MTHFD2 Inhibitor (DS18561882) with in Vivo Antitumor Activity.
J.Med.Chem., 62, 2019

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件を2024-07-17に公開中

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